Target Details
| UniProt AC | Q99814 |
|---|---|
| Gene Symbol | EPAS1 |
| Protein Name | Endothelial PAS domain-containing protein 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF23171 (bHLH_HIF1A) PF11413 (HIF-1) PF08778 (HIF-1a_CTAD) PF00989 (PAS) PF14598 (PAS_11) |
Summary
- Multi-target molecules 107
- Clinical molecules 0
- Avg pChEMBL 6.88
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (107)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RBKUARNZLBUCAG
|
6.7 | IC50 | 2 | — | |
BSLNBWGCFHYQTJ
|
6.6 | IC50 | 2 | — | |
BWSPDQARNUPHFS
|
6.6 | IC50 | 2 | — | |
CQGIUFASDNXPRB
|
6.5 | IC50 | 3 | — | |
FGDAZKGJPZGOKI
|
6.5 | IC50 | 2 | — | |
SRYXTPSNXWOGLW
|
6.5 | IC50 | 2 | — | |
JYXVAMLAJSGCDL
|
6.5 | IC50 | 2 | — | |
PCJSWXIBXCRFJH
|
6.5 | IC50 | 2 | — | |
IVWQWKFFMYQVHJ
|
6.5 | IC50 | 2 | — | |
WGJHLXZAYOERQG
|
6.5 | IC50 | 2 | — | |
ITVHGRMYDUEOHH
|
6.4 | IC50 | 2 | — | |
FBLSAINZUURAAQ
|
6.4 | Kd | 2 | — | |
CRDOBJXZSHDUKG
|
6.4 | IC50 | 2 | — | |
NKHJQIMZBYZZNI
|
6.4 | IC50 | 2 | — | |
BFZNXAFREFMQDF
|
6.4 | Kd | 2 | — | |
JTUWBMRONSWGPE
|
6.4 | IC50 | 2 | — | |
LTJZINXKULUVGF
|
6.4 | IC50 | 2 | — | |
PQZKMXPISWCLCU
|
6.4 | IC50 | 2 | — | |
ZPOVSMRTZGEMDG
|
6.4 | IC50 | 2 | — | |
QLSJHDNDYWPJFX
|
6.4 | IC50 | 2 | — | |
OGLFTTHUASEWEH
|
6.3 | IC50 | 2 | — | |
FYOFKDQRUFHOHF
|
6.3 | IC50 | 2 | — | |
BDRGEUHOAAKCOI
|
6.3 | IC50 | 2 | — | |
GJLPBJAKALWNPH
|
6.3 | Kd | 2 | — | |
QOIDRNFPRZOCJE
|
6.3 | IC50 | 2 | — | |
PBGRCXZQTHMAOP
|
6.3 | IC50 | 2 | — | |
FGCJEVWDLATQGD
|
6.3 | IC50 | 2 | — | |
MSLKJZNCDWDMHK
|
6.3 | Kd | 2 | — | |
XCTZRRRVHUREGM
|
6.3 | IC50 | 2 | — | |
ZOFBYPLMJZJZIK
|
6.2 | IC50 | 2 | — | |
AEDXHIJSHUQOIU
|
6.2 | IC50 | 2 | — | |
BJYORZAIOLJNDE
|
6.2 | IC50 | 2 | — | |
IPZJNJPAVPZHJM
|
6.2 | IC50 | 3 | — | |
DDQZGFIXHMUCKK
|
6.2 | IC50 | 2 | — | |
MSHAZOHWMOSOLX
|
6.2 | IC50 | 2 | — | |
SZZWTRXGNSPSOB
|
6.2 | IC50 | 2 | — | |
IRUDMTDFNXURLI
|
6.2 | Kd | 2 | — | |
DTBKRPGPPWHXPW
|
6.2 | IC50 | 2 | — | |
RBKUARNZLBUCAG
|
6.2 | IC50 | 2 | — | |
ZQVXDXKWSCKGBK
|
6.2 | IC50 | 2 | — | |
XNFHNRBWLZQXJI
|
6.2 | IC50 | 2 | — | |
DOHJEWQMMKPCDY
|
6.2 | IC50 | 2 | — | |
UEKZXQHSGGGLCW
|
6.2 | IC50 | 2 | — | |
WYHNPGCXYCAGNR
|
6.1 | IC50 | 2 | — | |
AHLKPENLDGAISD
|
6.1 | IC50 | 2 | — | |
XHJJPQRLFFDDTQ
|
6.1 | IC50 | 5 | — | |
XBLVKWKMJUNTSH
|
6.1 | IC50 | 2 | — | |
XWAGVAHGTLVLOU
|
6.1 | IC50 | 2 | — | |
MGNZDPRZMLYUEG
|
6.1 | IC50 | 2 | — | |
ADXGBBGMWKEJTR
|
6.0 | IC50 | 2 | — |