Target Details
| UniProt AC | Q99759 |
|---|---|
| Gene Symbol | MAP3K3 |
| Protein Name | Mitogen-activated protein kinase kinase kinase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00564 (PB1) PF00069 (Pkinase) |
Summary
- Multi-target molecules 26
- Clinical molecules 12
- Avg pChEMBL 6.82
KEGG Pathways (5)
Associated Diseases (1)
Active Molecules (26)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UIARLYUEJFELEN
|
8.2 | Kd | 289 | Yes | |
HKSZLNNOFSGOKW
|
8.0 | IC50 | 408 | — | |
MWKSRKSEWLRPBL
|
7.6 | Kd | 1075 | — | |
YRDHKIFCGOZTGD
|
7.5 | IC50 | 21 | — | |
XZXHXSATPCNXJR
|
7.5 | Kd | 165 | Yes | |
UBPYILGKFZZVDX
|
7.3 | Kd | 130 | Yes | |
KTEIFNKAUNYNJU
|
7.0 | Kd | 114 | — | |
YYLKKYCXAOBSRM
|
6.9 | Kd | 191 | — | |
JWNPDZNEKVCWMY
|
6.9 | Kd | 57 | Yes | |
HFNKQEVNSGCOJV
|
6.8 | Kd | 65 | — | |
NHHQJBCNYHBUSI
|
6.8 | Kd | 220 | — | |
ZCBUQCWBWNUWSU
|
6.8 | Kd | 59 | — | |
BMGQWWVMWDBQGC
|
6.7 | Kd | 147 | Yes | |
GUBJNPWVIUFSTR
|
6.7 | Kd | 103 | — | |
WINHZLLDWRZWRT
|
6.7 | Kd | 201 | Yes | |
RYYNGWLOYLRZLK
|
6.6 | Kd | 45 | — | |
ZBNZXTGUTAYRHI
|
6.5 | Kd | 102 | Yes | |
CTNPALGJUAXMMC
|
6.5 | Kd | 151 | — | |
QQWUGDVOUVUTOY
|
6.5 | Kd | 231 | Yes | |
LOLPPWBBNUVNQZ
|
6.5 | Kd | 97 | Yes | |
VAARYSWULJUGST
|
6.4 | Kd | 119 | Yes | |
DKZYXHCYPUVGAF
|
6.4 | Kd | 112 | — | |
CSGQVNMSRKWUSH
|
6.3 | Kd | 21 | — | |
MFAQYJIYDMLAIM
|
6.2 | Kd | 130 | Yes | |
YLCFOHVAOBLAIK
|
6.1 | IC50 | 14 | — | |
KGPGFQWBCSZGEL
|
6.1 | Kd | 59 | Yes |