Target Details
UniProt ACQ99720
Gene SymbolSIGMAR1
Protein NameSigma non-opioid intracellular receptor 1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF04622 (ERG2_Sigma1R)
Summary
  • Multi-target molecules 923
  • Clinical molecules 25
  • Avg pChEMBL 7.36
Top Co-occurrence Targets
Active Molecules (923)
InChIKey pChEMBL Type Targets Clinical
OUCUASFMBXPART 7.6 Ki 2
PBBXLWLZRSSICR 7.6 Ki 2
HQOMLTLQWBDVRA 7.6 Ki 2
DDIJOHSTGKDAKN 7.5 Ki 4
ORXZYLUNARJXOL 7.5 Ki 3
FDUWKETXXFSWBN 7.5 Ki 2
FSJMSQOSUBAJKA 7.5 Ki 2
HYJVYRBGCPGOSX 7.5 Ki 2
IWLWNPOFKPUZCM 7.5 Ki 2
LQPXVZLXNDSSPM 7.5 Ki 2
UEXJPFHGKCBUSS 7.5 Ki 3
FFCRKESJGXTNRJ 7.5 Ki 2
GREAMKHYUKBUBZ 7.5 Ki 2
JEYWNNAZDLFBFF 7.5 Ki 3
KVGNSDMVYWRLTG 7.5 Ki 10
UXMYQZAEDKKWCL 7.5 Ki 2
YSEXVIPNIGQQMN 7.5 Ki 5
CVRGNXKQUJMNME 7.5 Ki 2
IYFITMLPVWGURC 7.5 Ki 2
MNEDBWGEAFWGRR 7.5 Ki 3
MYNBCWZWZNXKKD 7.5 Ki 3
AOOSJYIINXVNHV 7.5 Ki 16
CAXQLHIXVZVOAJ 7.5 Ki 2
GFGDEBIFXMGQCV 7.5 Ki 3
IHGFBAKIGVPJDC 7.5 Ki 4
OMZGFFVAPHBNDW 7.5 Ki 2
OPNUROKCUBTKLF 7.5 Ki 2
PCWGGOVOEWHPMG 7.5 Ki 12
GOMIDUKJIYVMRM 7.5 Ki 3
LVXYAFNPMXCRJI 7.5 Ki 3
PSSRUTSUVLVFTJ 7.5 Ki 2
VBUAEXPIFRASGV 7.5 Ki 2
ADQJTHBSZROYBX 7.5 Ki 2
HYJVYRBGCPGOSX 7.5 Ki 2
LECUUDCCVOYUHG 7.5 Ki 7
OEILHFLXSQZBDT 7.5 Ki 2
BZGSLTDGENGQJF 7.5 Ki 3
IWOPGTFNUXEULQ 7.5 Ki 4
KRRIOBULVTVQLP 7.5 Ki 4
PHIVTHZDRRRWRB 7.5 Ki 2
STUOLNTZRBIDSI 7.5 Ki 2
WIKYUJGCLQQFNW 7.5 IC50 23 Yes
OKBJBWKATFFGNY 7.5 Ki 2
ARWONURFSGKTJW 7.4 Ki 7
CJOFXWAVKWHTFT 7.4 Ki 3
KFNBRURSYGJOHJ 7.4 Ki 3
NUYBPCYMEPUOQE 7.4 Ki 2
ACIKAIVCJBOQAN 7.4 Ki 3
AIDFXUXYEVBEFF 7.4 Ki 2
KWZTVVFHLUDCLT 7.4 Ki 2
2D structure