Target Details
UniProt ACQ99720
Gene SymbolSIGMAR1
Protein NameSigma non-opioid intracellular receptor 1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF04622 (ERG2_Sigma1R)
Summary
  • Multi-target molecules 923
  • Clinical molecules 25
  • Avg pChEMBL 7.36
Top Co-occurrence Targets
Active Molecules (923)
InChIKey pChEMBL Type Targets Clinical
KVOLGCQEWUQCJL 7.7 Ki 2
KVQVOBYCDUZJSF 7.7 Ki 2
SKCXLYQNMIOSKI 7.7 Ki 5
XRKKADYYRPDJSD 7.7 IC50 2
CFJMRBQWBDQYMK 7.7 Ki 4
CEMUKLXXZBFFNQ 7.7 Ki 2
DKNWSYNQZKUICI 7.7 Ki 2
KHQLKMURGRQDRK 7.7 Ki 2
LULSSQQQKPYPOR 7.7 Ki 2
OFAIGZWCDGNZGT 7.7 Ki 2
USTJOKQGVKRZCI 7.7 Ki 2
WEWQIJGSOWZYLM 7.7 Ki 2
HARWPKOPJYALIX 7.7 Ki 2
IBNDZHBEHXBGDO 7.7 Ki 2
OZRJHGKKLPXGID 7.7 Ki 2
RSVBTLSIVBWMNF 7.7 Ki 2
SQZBAUUHDXMUTO 7.7 Ki 4
VGBPBHGWCLWDSK 7.7 Ki 2
VYMHDKJVVMXTRF 7.7 Ki 2
HPZHSYBCGLDRCT 7.7 Ki 2
RSDAEFPWFADGBB 7.7 Ki 2
CBBXSFLTMNJOGU 7.7 Ki 5
CERLEBZSZWVJEJ 7.7 Ki 5
KZTQRGRPZOLMSL 7.7 Ki 3
RVMUAKCKCUJBKV 7.7 Ki 9
RZNGJRGWOYBVCK 7.7 Ki 3
SFPSQBFPUCFLEZ 7.7 Ki 9
YTWNFGCGMLTWHU 7.7 Ki 2
DKIOLBBRSOUKFN 7.6 Ki 2
JAKIOOTWQGBKAJ 7.6 Ki 2
KXRBNMSGFUSFLX 7.6 Ki 2
WFAJJUAIPMLRAE 7.6 Ki 2
YIJMQARSZOHNOV 7.6 Ki 2
BZSOPMPZSAMQIF 7.6 Ki 2
MVKKLGNVARQKRP 7.6 Ki 13
QVRVXSZKCXFBTE 7.6 Ki 2
QVRVXSZKCXFBTE 7.6 Ki 2
BXJUXLMPTUNFRY 7.6 Ki 2
MXKZBMGRCYCKSV 7.6 Ki 8
AUQCZPJCGAJBRC 7.6 Ki 4
DERZBLKQOCDDDZ 7.6 IC50 20 Yes
DTIGIZPIZLMRJY 7.6 Ki 2
IXSBEWUZWQANBY 7.6 Ki 2
KBEJBFGBZGNZHJ 7.6 Ki 2
PNANRXSVZAPWNF 7.6 Ki 5
YSSBJODGIYRAMI 7.6 Ki 2
ZEQHXVDOFWGIOA 7.6 Ki 5
CSHFTPUNJFOMTD 7.6 Ki 5
NKANXQFJJICGDU 7.6 Ki 35 Yes
NPAHFAYATIIHCN 7.6 Ki 2
2D structure