Target Details
UniProt ACQ99720
Gene SymbolSIGMAR1
Protein NameSigma non-opioid intracellular receptor 1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF04622 (ERG2_Sigma1R)
Summary
  • Multi-target molecules 923
  • Clinical molecules 25
  • Avg pChEMBL 7.36
Top Co-occurrence Targets
Active Molecules (923)
InChIKey pChEMBL Type Targets Clinical
PLDUPXSUYLZYBN 7.9 IC50 22
VAOKFJZCNXIHTK 7.9 Ki 2
PPZBZJPCFRFDCX 7.9 Ki 2
AJNXCTFYCKDBPU 7.8 IC50 8
AORIOLLAPPJVNF 7.8 Ki 2
BMUHJRCSESNQGV 7.8 Ki 3
KAPILGGLKCOQLO 7.8 Ki 2
QOXCLDKXSCBOOF 7.8 Ki 3
QXQOZVSPURYOAI 7.8 Ki 2
RSVBTLSIVBWMNF 7.8 Ki 3
SAPQZYMPGUOQOF 7.8 IC50 8
SGEGOXDYSFKCPT 7.8 Ki 18 Yes
ADEBPBSSDYVVLD 7.8 Ki 8
UAYVZHLRDFXTFC 7.8 Ki 2
WNZBBTJFOIOEMP 7.8 Ki 2
ADEBPBSSDYVVLD 7.8 Ki 6
BSLBJQNVSCZYMV 7.8 Ki 4
JRPGEMWAJXMXHL 7.8 Ki 2
ZEIMIZKOLIBIEH 7.8 Ki 3
ZEWQUBUPAILYHI 7.8 Ki 21
BCZGBRPOQMWWRA 7.8 Ki 2
FFCRKESJGXTNRJ 7.8 Ki 2
GTHHJVJOWMXRBS 7.8 Ki 3
HCXWPWPGUTZRDL 7.8 IC50 8
IKFBJNOEPLDTAT 7.8 Ki 9
JEAHRMVLQDOFBM 7.8 Ki 2
JYHPMRAWMPLJHU 7.8 Ki 2
SMANXXCATUTDDT 7.8 IC50 25 Yes
WLGVVEQIKFIUPU 7.8 Ki 3
XIQVNETUBQGFHX 7.8 IC50 10
YIVXLYPFIDEQFV 7.8 Kd 2
ZFQXVRJOHFYFDH 7.8 Kd 2
CJPSXNUMUGKDSS 7.8 Ki 2
DGPGXHRHNRYVDH 7.8 Ki 2
GLAFJHYUSDSQSZ 7.8 Ki 2
ITSKPCHXUYILTR 7.8 Ki 3
NHRNIDBKKUALMK 7.8 Ki 2
RAQPOZGWANIDQT 7.8 IC50 4
XWAONOGAGZNUSF 7.8 Ki 2
ZIDKNUHPKSUTKP 7.8 Ki 2
KZTINAFTXUOKGI 7.8 Ki 2
MFENLEFQLPLCJU 7.8 Ki 2
WGRSIFPGOSXXLA 7.8 Ki 2
CVCVHLAGPYEAKC 7.7 Ki 2
JMGCLJGEYSAHMV 7.7 Ki 4
MSYCGACUZCZLFO 7.7 Ki 2
XAOGFGMCKFYYEE 7.7 Ki 2
XSRZDWFALCQUFX 7.7 Ki 5
YTLYRBAXRSFIBF 7.7 Ki 2
IJLHWQBSZFONAR 7.7 Ki 2
2D structure