Target Details
UniProt ACQ99720
Gene SymbolSIGMAR1
Protein NameSigma non-opioid intracellular receptor 1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF04622 (ERG2_Sigma1R)
Summary
  • Multi-target molecules 923
  • Clinical molecules 25
  • Avg pChEMBL 7.36
Top Co-occurrence Targets
Active Molecules (923)
InChIKey pChEMBL Type Targets Clinical
FVMDOYQNOWAVCQ 8.4 Ki 5
MZEWTMVKHJXAGJ 8.4 Ki 2
SMBAOURHXAGUDO 8.4 Ki 2
FNQUSRALNJBLQF 8.4 Ki 2
FZTAXYPIZMGGRY 8.4 Ki 2
CRUMZXXYFKNNBD 8.4 Ki 2
XPPRDCVATUTJON 8.4 Ki 3
CYOAKAJZFCMXHY 8.4 Ki 2
DGIHILWHEUNSHI 8.4 Ki 2
SLJXLWDNADHNLA 8.4 Ki 2
UYNVMODNBIQBMV 8.4 IC50 10
UYNVMODNBIQBMV 8.4 IC50 5
DWAWDSVKAUWFHC 8.4 Ki 3
LQRUHPTVKTXHPR 8.4 Ki 2
NBNYXJWRMQPRPT 8.4 Ki 4
NTRXRHOREDBYQW 8.4 Ki 2
OWKPSSGANQPLEI 8.4 Ki 5
PFOHALKXQIXUFE 8.4 Ki 5
UMGDAMMXRYHVHZ 8.4 Ki 4
JUWUZLUBIRHYMM 8.4 Ki 3
LGSGJWDXMWVXEB 8.4 Ki 6
QSCBMVHTDSJVEE 8.4 Ki 3
AIHHKXSJJYAYND 8.4 Ki 2
CRUVUAJAFLBHLV 8.4 Ki 2
FKTFOSFQTJFKJX 8.4 Ki 2
YWPSNNQVCNRFAG 8.4 Ki 2
UVSWWUWQVAQPJR 8.4 Ki 2
UVSWWUWQVAQPJR 8.4 Ki 3
XKIGTQXAOLOQJD 8.4 Ki 4
AKFQMBJQZZAKNP 8.3 Ki 2
NTESFUMRHWXLJE 8.3 Ki 4
LPOOUTTZIAYDSP 8.3 Ki 2
BDECJFBHDUVJRU 8.3 Ki 6
YYCFTPUSYYQXNV 8.3 Ki 3
GKIRPKYJQBWNGO 8.3 Ki 4
PQUAPUMMXIRMPT 8.3 Ki 4
TXKBPYNMEJESGE 8.3 Ki 5
TYTUURCCMHKELI 8.3 Ki 5
DUUYHLUSDHATNS 8.3 Ki 3
JWNWVBYZLJCIIB 8.3 Ki 3
BXHPZOSDEOGGRA 8.3 Ki 2
HNGJYTQPOMPWSQ 8.3 Ki 2
JYSKWOSZRBRFQE 8.3 Ki 2
LVTANUBEUFAQCI 8.3 Ki 2
QLNOSQWPXXWXIP 8.3 Ki 2
ZNSPQQGMNDMVKM 8.3 Ki 2
DGDPBRUTRCRWFD 8.3 Ki 2
RHKLNFPODGBPGC 8.3 Ki 4
AKLDTUYECWDWIE 8.2 Ki 2
BXNNACCQTQBSOO 8.2 Ki 3
2D structure