Target Details
UniProt ACQ99720
Gene SymbolSIGMAR1
Protein NameSigma non-opioid intracellular receptor 1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF04622 (ERG2_Sigma1R)
Summary
  • Multi-target molecules 923
  • Clinical molecules 25
  • Avg pChEMBL 7.36
Top Co-occurrence Targets
Active Molecules (923)
InChIKey pChEMBL Type Targets Clinical
PMWDTSZFAMVNKX 8.8 Ki 2
VOKSWYLNZZRQPF 8.8 Ki 3
YUDTTWNDIWVWMJ 8.8 Ki 2
JCHUVGUKPFGRNQ 8.8 Ki 3
DGDSZKSHJGFASX 8.7 Ki 2
WNZBBTJFOIOEMP 8.7 Ki 2
CXMRZVOWSQPBGP 8.7 Ki 4
MBRMOGQHSBUGKH 8.7 Ki 2
QFTVLWSOZNQXAE 8.7 Ki 3
ZJUIXZLQJIZZJN 8.7 Ki 2
FVMIAKGRUAFNMJ 8.7 Ki 2
BNVHQFIRDRSKFK 8.7 Ki 2
FBWUQEIVZSYNQZ 8.7 Ki 5
JWSOZDLNDCOUIX 8.7 Ki 2
MYKJVLTXPNIGOV 8.7 Ki 2
UKBSDZLTDAZSCG 8.7 Ki 2
URDHIIFLGMSALF 8.7 Ki 4
UYNVMODNBIQBMV 8.7 Ki 8
BTEHVLUMUBTQOZ 8.7 Ki 3
IJKYJDDNDXAREJ 8.7 Ki 2
WWEAHUHMEHELLH 8.7 Ki 2
YEBCMFLMLQEJBU 8.7 Ki 2
WNZBBTJFOIOEMP 8.7 Ki 3
DEGAULWTOQJMMN 8.6 Ki 2
ZGKAPJYBJLXXMX 8.6 Ki 3
DICPGMOKBHQFRK 8.6 Ki 3
AEQDJSLRWYMAQI 8.6 Ki 2
YRTVIZSNPPJZLP 8.6 Ki 4
SQUNAWUMZGQQJD 8.6 IC50 2
BNRDJYCVXAIEIV 8.6 IC50 2
ADCBAOTWERXLAP 8.6 Ki 6
KRRIOBULVTVQLP 8.6 Ki 2
FHDBCFMWQMCVRI 8.5 Ki 2
NLEQSFUEJXECJY 8.5 Ki 7
VWZWORFVAMBTRI 8.5 Ki 2
HJJBGZORBJLFRB 8.5 Ki 2
LDSOWTPRMHWTOP 8.5 Ki 3
MLDCBJPLHBPJET 8.5 IC50 2
MYKJVLTXPNIGOV 8.5 Ki 3
UFVQFLZDNKHMBP 8.5 Ki 4
VOKSWYLNZZRQPF 8.5 Ki 4
CURUTKGFNZGFSE 8.5 IC50 10
TVEZSZAKGLHZOD 8.5 Ki 2
CPQKZLNBCUOHCW 8.5 Ki 3
SVALPNADURCFPN 8.5 Ki 2
IMFLKRNUSHCDBK 8.5 Ki 6
DXJUCAUQIHNOAF 8.5 IC50 2
LNEPOXFFQSENCJ 8.5 Ki 33 Yes
PCBKRGDPGXQWHV 8.5 Ki 2
DZKQLQVIZFRZDB 8.4 Ki 2
2D structure