Target Details
UniProt ACQ99720
Gene SymbolSIGMAR1
Protein NameSigma non-opioid intracellular receptor 1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF04622 (ERG2_Sigma1R)
Summary
  • Multi-target molecules 923
  • Clinical molecules 25
  • Avg pChEMBL 7.36
Top Co-occurrence Targets
Active Molecules (923)
InChIKey pChEMBL Type Targets Clinical
YMBWRCKWGRSBJG 6.5 Ki 2
HGRHWEAUHXYNNP 6.5 Ki 16
KTXMLKWFHNEBJM 6.5 Ki 2
YZSQCQQXQNXTIO 6.5 Ki 2
UPPMZCXMQRVMME 6.5 IC50 7
XPJMFYKZWMSEIT 6.5 Ki 2
YVIJCUAIMAKVQA 6.5 Ki 2
IYJQKAWJGMTUMA 6.5 Ki 2
KDOQEEMQPHIANX 6.5 Ki 2
NKJRGQRURURYMH 6.5 Ki 2
WJDLKMWEXVEBMK 6.5 Ki 9
SVJMLYUFVDMUHP 6.5 Ki 26
LFYNHAXLOHOWGV 6.5 Ki 2
PXWAOPCHLIOXQZ 6.5 IC50 7
CMWYFKYOUDIBBD 6.5 Ki 2
IBHQWHKVWRYMBH 6.5 Ki 2
MKXZASYAUGDDCJ 6.5 Ki 3
PQVQCEDGSJVHMK 6.5 Ki 9
GFIXZFAEEJIIGX 6.5 Ki 2
BZHBDEKYKFTCPD 6.4 Ki 2
DOMXUEMWDBAQBQ 6.4 IC50 3
DRSZMILOMUPIBJ 6.4 Ki 4
VQHIABNUZGYFSY 6.4 IC50 2
PHCDGYQTXVZSOO 6.4 Ki 2
HAZPAMUWUHDPDA 6.4 Ki 4
JWOJDKMHSKNBEA 6.4 Ki 3
LITALOXXZWFTOC 6.4 Ki 2
WKPMEBZKUOLVJC 6.4 Ki 2
YAVGJSSSBKISPN 6.4 Ki 2
BLJRIMJGRPQVNF 6.4 Ki 4
GOTMKOSCLKVOGG 6.4 IC50 9
HDDVHPLBIKYRCZ 6.4 Ki 2
OCAZOEMBQJUTFQ 6.4 Ki 2
BOOQTIHIKDDPRW 6.4 Ki 14
QTKHCKFFZZANPG 6.4 Ki 2
RNXYMZNGMNWKMC 6.4 Ki 3
XEPCAIUIHZEYAD 6.4 Ki 2
FJUKDAZEABGEIH 6.4 Ki 19
IILIVCVVZSPCRP 6.4 Ki 2
JXPQAZJMCCPVQL 6.4 Ki 2
KIGSHHDICVKMNF 6.4 Ki 2
ODQWQRRAPPTVAG 6.4 IC50 20 Yes
SWEOAXMICIJCQC 6.4 Ki 4
XTKDAFGWCDAMPY 6.4 Ki 8
DMEDHHKXKVEBDF 6.4 Ki 2
RIDKTDMXJSXQEJ 6.4 Ki 2
JUQLTPCYUFPYKE 6.4 Ki 25
JFHPNLALJKIFQH 6.4 Ki 2
DVYBIZHLZSDANU 6.3 Ki 4
DVYBIZHLZSDANU 6.3 Ki 2
2D structure