Target Details
UniProt ACQ99720
Gene SymbolSIGMAR1
Protein NameSigma non-opioid intracellular receptor 1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF04622 (ERG2_Sigma1R)
Summary
  • Multi-target molecules 923
  • Clinical molecules 25
  • Avg pChEMBL 7.36
Top Co-occurrence Targets
Active Molecules (923)
InChIKey pChEMBL Type Targets Clinical
QNOUNQTVKKLGSL 6.7 Ki 2
GYCXXEZMLXHNAI 6.7 Ki 2
QGQRUYNHBMRUGE 6.7 Ki 2
FVPJTKHMUKHCBG 6.7 Ki 2
OOGJQPCLVADCPB 6.7 Ki 9
WJLATVOFFJQTEJ 6.7 Ki 4
FCLQKBPRTZWHGX 6.7 Ki 2
JAQUASYNZVUNQP 6.7 IC50 8
OKBJBWKATFFGNY 6.7 Ki 2
WFLAIMWDHDADBE 6.7 Ki 2
TTWGDSSADVBNQY 6.7 Ki 12
NWJSAJQGUZTVMZ 6.6 Ki 2
PYSAVFUPLJMDHW 6.6 Ki 2
HTSNFXAICLXZMA 6.6 Ki 4
KLBQZWRITKRQQV 6.6 IC50 25 Yes
NFGZUZNICTWMFA 6.6 Ki 2
UFFHNEZNXKJHFB 6.6 Ki 10
ZPXSCAKFGYXMGA 6.6 IC50 4
ZPXSCAKFGYXMGA 6.6 IC50 4
ANFPJPBRQRWMFP 6.6 Ki 2
DOCRCBAANQJZLH 6.6 Ki 2
MCYCODJKXUJSAT 6.6 Ki 7
NFSPGABTRZUJES 6.6 Ki 2
POQDXIFVWVZVML 6.6 Ki 2
QWCRAEMEVRGPNT 6.6 IC50 12
UIQMVEYFGZJHCZ 6.6 IC50 4
DNKOFAGMIMGCMM 6.6 Ki 2
NWIUTZDMDHAVTP 6.6 Ki 3
NYQOWDCWPBGAEZ 6.6 Ki 2
CDDODAHZNGOHJP 6.6 Ki 2
GBFGNLHFJPHPAD 6.6 Ki 2
QXRFTZSLKJIIFB 6.6 Ki 4
FFCRKESJGXTNRJ 6.6 Ki 2
IPKSCZZHCDJCLO 6.6 Ki 2
MNHDKMDLOJSCGN 6.6 Ki 23
WSEQXVZVJXJVFP 6.6 IC50 6 Yes
DSEJCLDJIFTPPH 6.6 Ki 4
FITQSJBSXMDHOS 6.6 Ki 4
RDOIQAHITMMDAJ 6.6 Ki 13
RJKFOVLPORLFTN 6.6 Ki 10 Yes
JKPISQIIWUONPB 6.6 Ki 4
PHWBOXQYWZNQIN 6.6 IC50 6
PWXJESIQWPYCPX 6.6 Ki 2
QEHPEXFTPOUOLB 6.6 Ki 2
SGLYTKUAFQGFJG 6.6 Ki 2
SKMFMSUPYCIHLQ 6.5 Ki 2
IFOJFIZTMVVOCA 6.5 Ki 2
NRCUGEUXKFLUED 6.5 Ki 2
ZPEIMTDSQAKGNT 6.5 IC50 35 Yes
OAEWNSKRLBVVBV 6.5 Ki 3
2D structure