Target Details
UniProt ACQ99720
Gene SymbolSIGMAR1
Protein NameSigma non-opioid intracellular receptor 1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF04622 (ERG2_Sigma1R)
Summary
  • Multi-target molecules 923
  • Clinical molecules 25
  • Avg pChEMBL 7.36
Top Co-occurrence Targets
Active Molecules (923)
InChIKey pChEMBL Type Targets Clinical
ZRFIENOINCBMSZ 6.8 IC50 8
MBUVEWMHONZEQD 6.8 Ki 17 Yes
WVZYAHUNVJPRKP 6.8 Ki 2
XYJJFGCFMUCSKK 6.8 Ki 2
PXSPDEKPDFNBRT 6.8 Ki 2
VQJOLAVGGLHBJE 6.8 Ki 2
BTTOYOKCLDAHHO 6.8 Ki 10
CLWPAPPLOVGZLY 6.8 Ki 2
GMBNTSDGYBGPJD 6.8 Ki 2
LGQCVMYAEFTEFN 6.8 Ki 2
OABBIJYYEHSJIO 6.8 Ki 2
PDEWFHSOYCUZAW 6.8 Ki 4
GFOKIOIABHCPTK 6.8 Ki 5
VEZRZVARKZVJQE 6.8 Ki 2
ZUGPOQBHNCDHMW 6.8 Ki 2
AWIYLVWAILOVMX 6.8 Ki 10
DATRLTNBZWRBPI 6.8 Ki 12
OGAKLTJNUQRZJU 6.8 IC50 9
RYKGNRDBUCAXKP 6.8 Ki 2
IJYQIQINXOLXRB 6.8 Ki 2
QAFQNYQSHKJJPP 6.8 Ki 2
JLRVRJYCLBYOLO 6.8 Ki 2
PWBFOZFQIQJACN 6.8 Ki 2
RVPIRBSAJDVEMX 6.8 Ki 2
STXKDDCTHKRUNQ 6.8 Ki 2
ZLZAFQPDXYRKBT 6.8 Ki 2
AQRLDDAFYYAIJP 6.8 Ki 5
IKBKZGMPCYNSLU 6.8 Ki 13
HELVAYSYFPKPOV 6.7 Ki 2
KICAOHIBDYKDCJ 6.7 Ki 2
LVXYAFNPMXCRJI 6.7 Ki 3
PGGCRGAETLNAJC 6.7 Ki 11
RSUVYMGADVXGOU 6.7 IC50 4
VBONNDPACFTZMX 6.7 IC50 2
BUPHAKNPGZLFJL 6.7 Ki 2
JIRVELURMYQGKV 6.7 Ki 2
NJZKUBRAMHOLNY 6.7 Ki 2
AEUCUNJYBAAELI 6.7 Ki 2
DOOSVCDCTYOKQL 6.7 Ki 2
KKLZGWQBNXJWGZ 6.7 Ki 4
AGCJIQWBHFFGSG 6.7 Ki 2
DSIKQNYSFIESBM 6.7 Ki 2
HRYIDIDQOAKIIB 6.7 Ki 2
MYSZLXOHEWPTDC 6.7 Ki 2
RZXQAOZBWNZIHX 6.7 Ki 2
YVIJCUAIMAKVQA 6.7 Ki 2
GTABKUMYLUXCIH 6.7 Ki 7
JGCUFOXBUYJGBX 6.7 IC50 3
YPELFRMCRYSPKZ 6.7 IC50 9
GFMRIFXLIUPAFX 6.7 Ki 2
2D structure