Target Details
UniProt ACQ99720
Gene SymbolSIGMAR1
Protein NameSigma non-opioid intracellular receptor 1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF04622 (ERG2_Sigma1R)
Summary
  • Multi-target molecules 923
  • Clinical molecules 25
  • Avg pChEMBL 7.36
Top Co-occurrence Targets
Active Molecules (923)
InChIKey pChEMBL Type Targets Clinical
CCYRVZGWDNSBAQ 7.2 IC50 3
MNYSMGPLHSJGLY 7.2 Ki 2
NQDGCGNKNJWZHP 7.2 Ki 5
XMXHEBAFVSFQEX 7.2 IC50 17
NASMRBRQNLMHLZ 7.2 Ki 2
AGCJIQWBHFFGSG 7.2 Ki 2
FBFZJNQYPHJCAV 7.2 Ki 2
GTKJIRGLYALTCK 7.2 Ki 2
KKPMYWNQZNRGIK 7.2 IC50 5
LYZONYJDSRWDIH 7.2 Ki 2
MWLYNXDRIPHNJD 7.2 Ki 2
OBZZMDAWHDDOFN 7.2 Ki 2
XMHDSSGOIGKARI 7.2 Ki 2
YDJSSIDBMXCRMF 7.2 Ki 2
ZELXHOCJMVBKRQ 7.2 Ki 2
DDQBFKNOKOZBQK 7.2 Ki 2
DSGWSBURJGGYAE 7.2 Ki 2
DXUQNBORIUMGPM 7.2 Ki 2
FQZPTFIEUGPWMR 7.2 Ki 2
HWHLPVGTWGOCJO 7.2 IC50 6
MWIASLNTAGRGGA 7.2 Ki 6
NBTIJJVBAGEXFD 7.2 Ki 3
SNYFWQWLZIRNKD 7.2 Ki 2
SNYFWQWLZIRNKD 7.2 Ki 2
FSRWEIUCHHKGNY 7.2 Ki 2
OFSWDFDKUCDFDW 7.2 Ki 2
QOECKZUXJGSVMP 7.2 Ki 11
ZXZVSEDQEUIUHT 7.2 Ki 2
HTDIOUCPOHFDQH 7.1 Ki 14
JVKYZPBMZPJNAJ 7.1 Ki 2
MLUVEMSNRPMVHW 7.1 Ki 2
OSJJYEUEJRVVOD 7.1 IC50 17 Yes
SLEQRFMTAWGXRG 7.1 Ki 2
BFCDFTHTSVTWOG 7.1 IC50 11
CSWPKILRWGOCDB 7.1 Ki 2
FCUAEDWJSLQAOZ 7.1 Ki 2
FFOULWDEZZZKGY 7.1 Ki 2
HTSNFXAICLXZMA 7.1 IC50 4
KCNBAUKGODRNGM 7.1 IC50 8
YDJSSIDBMXCRMF 7.1 Ki 2
RCAWYRTWTRRNST 7.1 Ki 2
XHIUHIDIRNZTAW 7.1 Ki 7
WHTVZRBIWZFKQO 7.1 Ki 4
WHTVZRBIWZFKQO 7.1 Ki 5
MPWWGTFDWDZHRM 7.1 Ki 10
PBFDUYRSNDQIDN 7.1 Ki 13
TYIUBVMXOWXQTD 7.1 Ki 2
XYNPYHXGMWJBLV 7.1 Ki 3
ZJAXDNQQFMPNAV 7.1 Ki 5
ZMDOBTILJRLEOG 7.1 Ki 3
2D structure