Target Details
UniProt ACQ99720
Gene SymbolSIGMAR1
Protein NameSigma non-opioid intracellular receptor 1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF04622 (ERG2_Sigma1R)
Summary
  • Multi-target molecules 923
  • Clinical molecules 25
  • Avg pChEMBL 7.36
Top Co-occurrence Targets
Active Molecules (923)
InChIKey pChEMBL Type Targets Clinical
GQNSENQYHXKTOP 7.3 Ki 2
RHMYPZYXJBYMPC 7.3 Ki 2
VBUAEXPIFRASGV 7.3 Ki 2
BKSVBMZEXVBOKL 7.3 Ki 2
BTJSYOUOQORWBA 7.3 Ki 4
CPJJMPKJBZZIIY 7.3 Ki 2
DFNAAFSXZVGDBJ 7.3 Ki 6
PFOWCBUJJWGNHA 7.3 Ki 2
PGALYKJJGGBYSX 7.3 Ki 2
QPMLJPMWNURBDC 7.3 Ki 2
SPOWGSLLJYGDKG 7.3 Ki 2
SYHLJLZHXZVWRS 7.3 Ki 2
ZZJYIKPMDIWRSN 7.3 IC50 8
DWWWTAMWZKMEOL 7.3 Ki 2
HBIVMNLRHOPKEJ 7.3 Ki 2
HBOJWAYLSJLULG 7.3 Ki 5
NWICMXBOJMLOIB 7.3 Ki 3
QVSZFVNYJYNUGG 7.3 Ki 2
WPFUJFQBOHAMPJ 7.3 Ki 2
GUJRSXAPGDDABA 7.3 Ki 4
QMZYZVGBMAHPDU 7.3 Ki 2
SVTYKQJVCXBJNT 7.3 Ki 2
ZBXIRNVCPMZPFS 7.3 Ki 2
RGHKOAFUHZEYJM 7.2 Ki 4
UYQJQXBCVBDUGX 7.2 Ki 2
BZPKTOXVMUIFBK 7.2 Ki 2
DHIDSSXNRVGMDP 7.2 Ki 2
LVWSRFJAMQNXCY 7.2 Ki 2
QHLAPIQLWATZKM 7.2 Ki 12
QNSPFRSAEHVDGL 7.2 Ki 4
VGKDLMBJGBXTGI 7.2 Ki 15
WWLFCQLHCAEMAP 7.2 Ki 4
MEKSQRMXWZHFIP 7.2 Ki 13
RIAXXCQKICATHW 7.2 IC50 8
VMJYYMFCJIJUTA 7.2 Ki 2
ZTXUPPVTVPOTMG 7.2 Ki 2
GJDLVCLPWHWXGI 7.2 Ki 2
INGWKGCHJJYQIB 7.2 IC50 3
ZDZZHGWPDPCPMZ 7.2 Ki 2
BWXABDUNWUIBLQ 7.2 Ki 3
HPMFKLUVLCAJPU 7.2 Ki 2
INCPDVXLHDEOLM 7.2 Ki 2
VFTROENQUWUAES 7.2 Ki 2
GUOJTYBMIRVPKO 7.2 Ki 2
ISQAPFMBJFZOLG 7.2 Ki 2
KRUXANLFCJDAMX 7.2 Ki 2
LYDQCJJNPZBLSS 7.2 Ki 2
SXDNKQKMHDBAAG 7.2 Ki 3
TUSPVTWVRDALHT 7.2 Ki 7
YZWJNFUQGOYUQT 7.2 Ki 7
2D structure