Target Details
UniProt ACQ99720
Gene SymbolSIGMAR1
Protein NameSigma non-opioid intracellular receptor 1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF04622 (ERG2_Sigma1R)
Summary
  • Multi-target molecules 923
  • Clinical molecules 25
  • Avg pChEMBL 7.36
Top Co-occurrence Targets
Active Molecules (923)
InChIKey pChEMBL Type Targets Clinical
DNGYIBDXSUNKMV 11.6 Ki 2
QEHXWPHILAGKIT 10.9 Ki 2
RTSYUWSEYYHQLC 10.5 Ki 2
YTOPFCCWCSOHFV 10.4 Ki 3
RYAUSSKQMZRMAI 10.1 Ki 3
YNZFUWZUGRBMHL 9.7 Ki 3
PJMPHNIQZUBGLI 9.4 Ki 6
FOQRKFCLRMMKAT 9.4 Ki 2
AINAOXBEBHZWSP 9.3 Ki 3
SPCBJRRRNGZOBD 9.3 Ki 2
YSACNAXEZHCMEQ 9.3 Ki 3
DXJUCAUQIHNOAF 9.3 IC50 6
QOXCLDKXSCBOOF 9.2 Ki 3
FPSFVONLLBIZFK 9.2 Ki 2
LDFPQKADFLEDQV 9.2 Ki 5
ILMRWZKEGUJTGG 9.2 Ki 2
SXWSMORDUABOEW 9.2 Ki 2
SMEIMTHKRVPONN 9.1 Ki 2
XBLBQWNQIGPMRE 9.1 Ki 2
GPMXUUPHFNMNDH 9.1 Ki 4
GWZNBTHONPZRPP 9.1 IC50 3
NNACHAUCXXVJSP 9.0 Ki 4
VWIJXNRUNDGWHS 9.0 Ki 2
HRBKFQYSVXXYDE 9.0 Ki 2
AJZBPCAHQHCXMX 9.0 Ki 5
DMZCCFMMPHJWQY 9.0 Ki 3
DWAWDSVKAUWFHC 9.0 Ki 3
FPCCSQOGAWCVBH 9.0 IC50 16
HOPPBDCZOOMPDL 9.0 Ki 2
KLBJRPVUPJXXCM 9.0 Ki 3
WMBHBWPQFUUUCP 9.0 Ki 4
BJMSSYYAXURYLB 9.0 Ki 2
KOYQYIAABUPJFF 9.0 Ki 2
FNNNBFYNDLVVGH 8.9 Ki 2
PZWPPSAANHYITK 8.9 Ki 4
XBTOAGKXNKAIIR 8.9 Ki 2
YBLIQJGXRLZBCZ 8.9 IC50 3
YMUGOAUDWIAQBS 8.9 Ki 2
VVPJKZNOOONNDJ 8.9 Ki 3
YBHXONPJHWVDCG 8.9 Ki 2
ZBAJQMFEBGHQTH 8.9 Ki 2
HLNYWGVTKKMJCB 8.8 Ki 2
KTHLRNWGDXCNQL 8.8 Ki 2
SACMWQXEALUQNE 8.8 Ki 2
RTCBVXFDQGRSDA 8.8 Ki 3
CPJJVXHVUGIXFK 8.8 Ki 2
PXJRNSSFQSUUFC 8.8 Ki 2
XQIPLSFFYJNKFR 8.8 Ki 2
ZVTTUTCRXOMKJP 8.8 Ki 2
HELCSESNNDZLFM 8.8 Ki 2
2D structure