Target Details
| UniProt AC | Q99705 |
|---|---|
| Gene Symbol | MCHR1 |
| Protein Name | Melanin-concentrating hormone receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 285
- Clinical molecules 6
- Avg pChEMBL 7.73
KEGG Pathways (2)
Active Molecules (285)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZYFROZAPTFMWIE
|
6.8 | IC50 | 2 | — | |
UGWKDYRCSUMLFR
|
6.7 | IC50 | 2 | — | |
XFYUYPSWQGVSKG
|
6.7 | IC50 | 2 | — | |
COLOFELGEFWPSM
|
6.7 | IC50 | 2 | — | |
RRWCFKTVVCKJCF
|
6.7 | Ki | 2 | — | |
WBVAZKKBRDFWSE
|
6.6 | Ki | 2 | — | |
GTMASPVXPKDKOK
|
6.6 | Ki | 3 | — | |
RDTRAPTXBPRALK
|
6.6 | Ki | 2 | — | |
AUHFSEIMAYONHH
|
6.6 | IC50 | 2 | — | |
KOMGNGDDTPNSKC
|
6.6 | Ki | 3 | — | |
DFSPHRXFDNSOGP
|
6.6 | IC50 | 2 | — | |
ZLLOVWBBACAVIV
|
6.5 | Ki | 3 | — | |
JHYBPHVVKVPUAR
|
6.5 | IC50 | 2 | — | |
FFRCQBGVCKTCAM
|
6.5 | IC50 | 2 | — | |
WHABNFKDVVGXEU
|
6.5 | Ki | 2 | — | |
RDLXVBBHIFGTEH
|
6.5 | Ki | 2 | — | |
QWVFLOZCIRVGKF
|
6.4 | Ki | 2 | — | |
OFKFNGSBLPQTPU
|
6.4 | IC50 | 2 | — | |
OWVJFLOWTRTEOY
|
6.3 | Ki | 2 | — | |
AKAAKXSPGNFTCK
|
6.3 | Ki | 2 | — | |
XQPIUMZQPPLXSB
|
6.3 | IC50 | 2 | — | |
KWGDXCJEWFIBAA
|
6.2 | Ki | 2 | — | |
BEWRGASHJMEIJG
|
6.2 | IC50 | 3 | — | |
SHSVOLDXXBHQPQ
|
6.2 | IC50 | 2 | — | |
RZFIMUGJIHXZIF
|
6.2 | IC50 | 2 | — | |
KJCQYSICJWKIHX
|
6.2 | IC50 | 2 | — | |
BOAIJXQJMLWMSF
|
6.2 | Ki | 3 | — | |
YHHIHIHYYOQBLJ
|
6.1 | IC50 | 2 | — | |
SXUROQLTGFUQFZ
|
6.1 | IC50 | 2 | — | |
RYUJZKYTNJACIJ
|
6.1 | IC50 | 3 | — | |
BOAIJXQJMLWMSF
|
6.1 | Ki | 3 | — | |
VSACRBUHJYUONF
|
6.1 | IC50 | 2 | — | |
CQEKVDIALJJBIO
|
6.0 | IC50 | 2 | — | |
PNEQLTWPDVHRRF
|
6.0 | IC50 | 3 | — | |
UGTJLUOFSLGNDT
|
6.0 | IC50 | 3 | — |