Target Details
| UniProt AC | Q99705 |
|---|---|
| Gene Symbol | MCHR1 |
| Protein Name | Melanin-concentrating hormone receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 285
- Clinical molecules 6
- Avg pChEMBL 7.73
KEGG Pathways (2)
Active Molecules (285)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SPPVYRMMRKTURF
|
7.3 | IC50 | 2 | — | |
LXGKPUINNMCWKV
|
7.3 | IC50 | 2 | — | |
GGPDSNHLDADOIF
|
7.2 | IC50 | 2 | — | |
OKIVGPUCUWMOIH
|
7.2 | IC50 | 3 | — | |
AZXDIBWQNPKWII
|
7.2 | Ki | 2 | — | |
NKKHUNXEXXFYQF
|
7.2 | IC50 | 2 | — | |
RRTFGNWCQSMHSP
|
7.2 | IC50 | 2 | — | |
AVSZXIJMFUSBBN
|
7.2 | Ki | 2 | — | |
HHCYCBKPWYJVEB
|
7.2 | IC50 | 3 | — | |
SNIGHIUCPHRJBN
|
7.2 | Ki | 2 | — | |
CPSZHSLGOIQVNS
|
7.2 | Ki | 2 | — | |
HKBQLXYNZOLAHS
|
7.2 | IC50 | 2 | — | |
ASKSJOULXJIZKH
|
7.2 | Ki | 2 | — | |
MHZCWVOMNJUVMC
|
7.1 | IC50 | 2 | — | |
INNDGUNGHHCVFO
|
7.1 | IC50 | 2 | — | |
VJPTYAZXVBTBPT
|
7.1 | IC50 | 2 | — | |
JJQLRTKUCLCIPR
|
7.1 | IC50 | 3 | — | |
LDCMGLYXOOMRFQ
|
7.1 | IC50 | 3 | — | |
ZTFJHOQHIJEDFE
|
7.1 | Ki | 2 | — | |
MHPRRIFCBPETQG
|
7.0 | IC50 | 3 | — | |
LLWKBGRAWPNWFD
|
7.0 | IC50 | 2 | — | |
SWOGBCMCJSXRTN
|
7.0 | IC50 | 2 | — | |
YECSPBDBORKKPX
|
7.0 | IC50 | 2 | — | |
AIDALYBWFLHEJP
|
7.0 | IC50 | 2 | — | |
UDROTHQORZMMBF
|
7.0 | IC50 | 2 | — | |
IZLJKNPYMLZCPG
|
7.0 | IC50 | 2 | — | |
NFQWOMAFZMZYOX
|
6.9 | IC50 | 5 | Yes | |
NQWRDTGSEHHGJT
|
6.9 | Ki | 2 | — | |
SUYDUGVDUFCDHQ
|
6.9 | Ki | 3 | — | |
GKDBTHSYQZTDAJ
|
6.9 | IC50 | 13 | — | |
IHXFHHOZRJEQBX
|
6.9 | IC50 | 2 | — | |
SUYDUGVDUFCDHQ
|
6.9 | Ki | 3 | — | |
FSTDLRINZOKGRA
|
6.9 | Ki | 3 | — | |
GPEOXJGBWGMANI
|
6.8 | IC50 | 3 | — | |
NJWKXGIQDOFDKH
|
6.8 | IC50 | 3 | — | |
CAIOOXOPQUHZGS
|
6.8 | Ki | 2 | — | |
RASPHJGGIPBIMT
|
6.8 | IC50 | 2 | — | |
JGSWRBZQDGUIET
|
6.8 | IC50 | 2 | — | |
SPZVGUOPAIQFIW
|
6.8 | IC50 | 2 | — | |
ZZCFQOGPJUCWRJ
|
6.8 | IC50 | 2 | — | |
HYNXKHHGAXLIEQ
|
6.8 | Ki | 3 | — | |
NTZDCPIPBYWRFF
|
6.8 | IC50 | 2 | — | |
NWUCPBLQECHRFK
|
6.8 | IC50 | 3 | — | |
NWUCPBLQECHRFK
|
6.8 | IC50 | 3 | — | |
PAXJABBAIBFJBH
|
6.8 | Ki | 4 | — | |
WTVQMTFZYWXSRS
|
6.8 | Ki | 4 | — | |
BHEGDYSAYYZJGP
|
6.8 | IC50 | 2 | — | |
KIOITPZEEHNURK
|
6.8 | IC50 | 2 | — | |
STDVLBNQKXFBHQ
|
6.8 | Ki | 2 | — | |
DOYKZJFYZSSDTP
|
6.8 | IC50 | 2 | — |