Target Details
| UniProt AC | Q99705 |
|---|---|
| Gene Symbol | MCHR1 |
| Protein Name | Melanin-concentrating hormone receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 285
- Clinical molecules 6
- Avg pChEMBL 7.73
KEGG Pathways (2)
Active Molecules (285)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JTXZPQNLRJKZDT
|
7.8 | IC50 | 2 | — | |
HLRRHIITKGDLDO
|
7.8 | IC50 | 2 | — | |
PHCHRPWAMGPRTQ
|
7.8 | IC50 | 2 | — | |
VWGMHCJKUIOSFN
|
7.8 | IC50 | 2 | — | |
HPMOYSAWXGTKNO
|
7.7 | IC50 | 2 | — | |
KLVCXDDJHLESAO
|
7.7 | IC50 | 2 | — | |
KTNRAOBLSVMKID
|
7.7 | IC50 | 2 | — | |
UKBMUBRWLVXPNM
|
7.7 | IC50 | 2 | — | |
GOGGRAWNDKPWNO
|
7.7 | IC50 | 2 | — | |
SQORIUUNRIGPKO
|
7.7 | IC50 | 2 | — | |
HJXJZSZXJNHUQH
|
7.7 | IC50 | 2 | — | |
CFIVGUWEJMEWCY
|
7.7 | IC50 | 2 | — | |
XLHNDXFCDIKZCH
|
7.7 | Ki | 2 | — | |
YNFBUKHNBHSFFK
|
7.7 | IC50 | 2 | — | |
KNFCUBWPKYSSNK
|
7.7 | IC50 | 2 | — | |
KGFPROOGUUWDFD
|
7.7 | IC50 | 2 | — | |
KXJVMFXTTSRQMV
|
7.7 | IC50 | 2 | — | |
IHNSUBDSHNRLFA
|
7.6 | IC50 | 2 | — | |
QDLQBKBQLRPJEG
|
7.6 | IC50 | 2 | — | |
QOKHHPNTBNJONY
|
7.6 | Ki | 2 | — | |
BXZRDVSRUIVYLG
|
7.6 | Ki | 2 | — | |
VMFNUQHBZCMQRZ
|
7.6 | IC50 | 2 | — | |
LXFOFQVESUDTGV
|
7.6 | Ki | 2 | — | |
PFTYUXPUTSSSAS
|
7.6 | IC50 | 2 | — | |
WQBXCEPRRLBKSC
|
7.6 | IC50 | 2 | — | |
BKKPIQPFRAPEAY
|
7.6 | IC50 | 2 | — | |
NZXNWHUQQIMGJQ
|
7.6 | Ki | 2 | — | |
GIAMAPLWLDNOGA
|
7.5 | IC50 | 2 | — | |
UGDQKRGYVYUTTP
|
7.5 | IC50 | 2 | — | |
SCBFPLDUOJGCDI
|
7.5 | IC50 | 2 | — | |
RZJWWQSGWHXWAK
|
7.5 | Ki | 2 | — | |
UQBHXZLKMLKWPT
|
7.5 | IC50 | 2 | — | |
PUTAQVRRQAPAQX
|
7.5 | IC50 | 2 | — | |
MZNNAIHCWWROJM
|
7.4 | IC50 | 2 | — | |
OLOYPXPKAJGIQP
|
7.4 | IC50 | 2 | — | |
JJZSKQSMTGTKID
|
7.4 | IC50 | 2 | — | |
RAUHDNCAWVVITH
|
7.4 | IC50 | 2 | — | |
VDTTVUDVHKAPMC
|
7.4 | IC50 | 3 | — | |
VMMGFPNGNCDEDD
|
7.4 | IC50 | 2 | — | |
XLARMCNJVYOFFY
|
7.4 | IC50 | 2 | — | |
KWMMLXRVWDEIDY
|
7.4 | IC50 | 2 | — | |
PYGPEGZKDLTLHJ
|
7.4 | IC50 | 2 | — | |
LNBYGAAFTSNLNC
|
7.4 | Ki | 2 | — | |
XUBSUXYAIPDFRU
|
7.4 | IC50 | 2 | — | |
FLYSTSPNPXBSFJ
|
7.4 | Ki | 2 | — | |
QQQVMCCARMEQHB
|
7.3 | Ki | 2 | — | |
QNCNYSGUYPUZKJ
|
7.3 | IC50 | 2 | — | |
WIFGAYBFSSWCPA
|
7.3 | Ki | 2 | — | |
AMVUYMPRVIDZMG
|
7.3 | IC50 | 2 | — | |
YHVMAQQCYJWINX
|
7.3 | IC50 | 2 | — |