Target Details
| UniProt AC | Q99705 |
|---|---|
| Gene Symbol | MCHR1 |
| Protein Name | Melanin-concentrating hormone receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 285
- Clinical molecules 6
- Avg pChEMBL 7.73
KEGG Pathways (2)
Active Molecules (285)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FAIMGWSOSCFGRU
|
8.1 | IC50 | 6 | Yes | |
AIVCREQIHBXHNV
|
8.1 | IC50 | 2 | — | |
CCQQMKPBDIACQQ
|
8.1 | IC50 | 2 | — | |
BWWACMBLBNGFJZ
|
8.1 | IC50 | 2 | — | |
YHSRTUXPXLVIAG
|
8.1 | IC50 | 3 | Yes | |
ZRXFYRUEDDMFHH
|
8.1 | Ki | 2 | — | |
ZITSWKKGCZZGDB
|
8.1 | IC50 | 2 | — | |
LOVAEQYMKDVCHF
|
8.0 | IC50 | 2 | — | |
FWSBSBDRADXORX
|
8.0 | IC50 | 2 | — | |
ZICGUURZNAJJKQ
|
8.0 | IC50 | 2 | — | |
DDSVEFMFCAHZEM
|
8.0 | IC50 | 2 | — | |
IESRGXWBZDJPLC
|
8.0 | IC50 | 2 | — | |
QJVKSHKJQIYIKU
|
8.0 | IC50 | 2 | — | |
JNOSYXLLGUQJNO
|
8.0 | IC50 | 2 | — | |
LNOMHNHLGYHPNB
|
8.0 | IC50 | 2 | — | |
OCMCRRBEHXHBIV
|
8.0 | IC50 | 2 | — | |
SNBBROUTMGTRAU
|
8.0 | IC50 | 2 | — | |
XEOSDWIUBUJPES
|
8.0 | IC50 | 3 | — | |
CYYAXTCZGPRATM
|
8.0 | IC50 | 2 | — | |
MCXDOOMLRVVNIJ
|
8.0 | IC50 | 2 | — | |
YHMGBTHOLTYBSS
|
8.0 | IC50 | 2 | — | |
BLVUILRZDGFJPZ
|
8.0 | IC50 | 2 | — | |
LCXRMOKMNODMLL
|
8.0 | IC50 | 2 | — | |
TUISOQBOQRFWFJ
|
8.0 | IC50 | 2 | — | |
ZZUJEMNDSKZYLV
|
8.0 | IC50 | 2 | — | |
MQEGXNOOYXGZRV
|
8.0 | Ki | 2 | — | |
RKFUUDHVACYQEP
|
8.0 | Ki | 2 | — | |
RRRMNLLTGSQHGV
|
7.9 | IC50 | 2 | — | |
DOKSQMPMAHUKLJ
|
7.9 | Ki | 2 | — | |
GXZNBYLIQYWZLV
|
7.9 | IC50 | 2 | — | |
OHLRSGMODYTCJK
|
7.9 | IC50 | 2 | — | |
BZNSXKFFBJLSJV
|
7.9 | IC50 | 2 | — | |
BZUVXLPHVGFEJA
|
7.9 | IC50 | 2 | — | |
CMNAXSCFAFPUGW
|
7.9 | IC50 | 2 | — | |
NDWXGJDJKXDMOV
|
7.9 | IC50 | 3 | — | |
ZMJZGADTCFELGA
|
7.9 | Ki | 2 | — | |
ZZOFPJLORHEXGT
|
7.9 | IC50 | 2 | — | |
TWNPKIQHYYMCGF
|
7.9 | IC50 | 2 | — | |
PGRNXALRNBGGDQ
|
7.8 | IC50 | 2 | — | |
RWHIDQWJRLHVCH
|
7.8 | IC50 | 2 | — | |
BXGRLXRXUOGKTC
|
7.8 | IC50 | 2 | — | |
KURYMMXNUSXWIX
|
7.8 | IC50 | 2 | — | |
MZYXOMZPGDOVJK
|
7.8 | IC50 | 2 | — | |
WGXXTIHJEXZLJF
|
7.8 | IC50 | 2 | — | |
MXDHYBKFGPNDFR
|
7.8 | IC50 | 2 | — | |
FWKVXHBRMCTKHZ
|
7.8 | Ki | 2 | — | |
GALAIUNXQRYFIW
|
7.8 | IC50 | 2 | — | |
HSFWTAVXXXJJRW
|
7.8 | IC50 | 2 | — | |
JCSAJCBJJWFNIO
|
7.8 | IC50 | 5 | Yes | |
GJOARULBWVWENP
|
7.8 | IC50 | 2 | — |