Target Details
| UniProt AC | Q99705 |
|---|---|
| Gene Symbol | MCHR1 |
| Protein Name | Melanin-concentrating hormone receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 285
- Clinical molecules 6
- Avg pChEMBL 7.73
KEGG Pathways (2)
Active Molecules (285)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IRTFNVYFUVVXDO
|
8.4 | IC50 | 2 | — | |
MGBCOVVRZAHNAM
|
8.4 | IC50 | 2 | — | |
VHNFRNTVRLAIBR
|
8.4 | IC50 | 2 | — | |
GIUYGLISRAEYOJ
|
8.4 | Ki | 2 | — | |
HWSUJLBBZVSJFM
|
8.4 | Ki | 3 | — | |
MABBTFRQYAXJAE
|
8.4 | IC50 | 2 | — | |
MQOANKATOVPZEV
|
8.4 | IC50 | 2 | — | |
ODSPZLQLPQOLJR
|
8.4 | IC50 | 3 | — | |
SZJOZHJPOSHWMC
|
8.4 | IC50 | 2 | — | |
TVRSQRQEYMGJLM
|
8.4 | IC50 | 2 | — | |
ZOKQZJZIENINDP
|
8.4 | IC50 | 2 | — | |
LSDCVVODSBVDMA
|
8.4 | IC50 | 2 | — | |
WDZOVHZBQNDKJX
|
8.4 | IC50 | 2 | — | |
PCMKFHUKCPUDQK
|
8.3 | IC50 | 2 | — | |
KTRMFSXYMXPKHJ
|
8.3 | IC50 | 2 | — | |
XJARKGGVDJGJMK
|
8.3 | IC50 | 2 | — | |
VVRXCUBJCBJGHR
|
8.3 | Ki | 2 | — | |
HZPGVFKYDDQWIZ
|
8.3 | IC50 | 4 | — | |
JLBZQGVJKAWCSE
|
8.3 | IC50 | 2 | — | |
ODLVSMAEEPBMLK
|
8.3 | IC50 | 2 | — | |
XKVMOBBNFSXUMW
|
8.3 | IC50 | 2 | — | |
ARFXECJNWZZFLK
|
8.3 | IC50 | 2 | — | |
BMVVLXNEZZJMOQ
|
8.3 | IC50 | 2 | — | |
JQTAYQKKSGXRPR
|
8.3 | IC50 | 2 | — | |
KLPGSSBKQHEWRL
|
8.3 | IC50 | 2 | — | |
KWGHMJGFVYVORH
|
8.3 | IC50 | 2 | — | |
OOUPDYBXVFKJRL
|
8.3 | IC50 | 2 | — | |
QHRSOSACJBYXIL
|
8.3 | IC50 | 2 | — | |
UGUPGQUFTPDBTH
|
8.3 | IC50 | 2 | — | |
WDEKEIWPPYORJF
|
8.3 | Ki | 2 | — | |
ANCFKYJMXNMYNZ
|
8.2 | IC50 | 3 | — | |
KESABOVUGAHUQM
|
8.2 | IC50 | 2 | — | |
RMXXLBXAQDDMHW
|
8.2 | IC50 | 2 | — | |
JFKJLEGVSYQSFA
|
8.2 | IC50 | 2 | — | |
RFTNZWFCHDUSMZ
|
8.2 | IC50 | 2 | — | |
BAZQBEOFVYAFHT
|
8.2 | IC50 | 5 | Yes | |
ZGQSHOMCFXQQCY
|
8.2 | IC50 | 2 | — | |
HTPPRDGEOSXUGA
|
8.2 | IC50 | 2 | — | |
WLBXFMNETGMZFI
|
8.2 | IC50 | 2 | — | |
CIMJGOFPRRZLKM
|
8.2 | IC50 | 2 | — | |
CYJMDICCNHFYPK
|
8.2 | IC50 | 2 | — | |
GFECAWJPCXIEEK
|
8.2 | Ki | 2 | — | |
SHCFFLWIRMAQPN
|
8.2 | IC50 | 2 | — | |
ZKAMUYRESJQUBC
|
8.2 | IC50 | 3 | — | |
HDLPZLIRDMOMBU
|
8.2 | Ki | 3 | — | |
INKLXDAZBDXKOH
|
8.2 | IC50 | 2 | — | |
ROIFDGZSVAMLHB
|
8.2 | IC50 | 2 | — | |
UKHHETYTQCSWPT
|
8.2 | IC50 | 2 | — | |
XKNDXALUSFQZAX
|
8.2 | IC50 | 3 | — | |
ZLKBWMPLNFUMFD
|
8.2 | IC50 | 2 | — |