Target Details
| UniProt AC | Q99705 |
|---|---|
| Gene Symbol | MCHR1 |
| Protein Name | Melanin-concentrating hormone receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 285
- Clinical molecules 6
- Avg pChEMBL 7.73
KEGG Pathways (2)
Active Molecules (285)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WNKKIZAQIDNXQY
|
10.5 | Ki | 2 | — | |
CTNRLCXTSKIWEA
|
9.9 | IC50 | 2 | — | |
JTNZOYWLPSIJGI
|
9.8 | Ki | 2 | — | |
GOKWVWMOVLFRQZ
|
9.7 | IC50 | 2 | — | |
CFUPTNNNCZABDF
|
9.6 | IC50 | 2 | — | |
OIWNBHQIKDINGT
|
9.5 | Ki | 2 | — | |
TUIRYRPRPHCOOR
|
9.4 | Ki | 3 | — | |
ZECBAHZJBRDQQI
|
9.4 | Ki | 2 | — | |
OXFHENXEDBVILO
|
9.3 | Ki | 2 | — | |
GUSAOPYZFQQULB
|
9.2 | IC50 | 2 | — | |
DJTVQVIZMNHBCR
|
9.0 | IC50 | 2 | — | |
IOVSXXYNGKBAID
|
9.0 | IC50 | 2 | — | |
OKJKIOJUDZFVDL
|
9.0 | IC50 | 2 | — | |
CFUPTNNNCZABDF
|
8.9 | IC50 | 2 | — | |
IYEJAIHDFCXVRY
|
8.9 | IC50 | 2 | — | |
FWMHZWMPUWAUPL
|
8.9 | IC50 | 2 | — | |
OMZPZOSWJGZBRV
|
8.8 | IC50 | 2 | — | |
RRZYXZCEHAPBIS
|
8.8 | IC50 | 2 | — | |
FBFVVUFMHULKRE
|
8.8 | IC50 | 2 | — | |
YWHDVYSFGAWVFS
|
8.7 | Ki | 2 | — | |
FTXAKSJEBVGKHR
|
8.7 | IC50 | 2 | — | |
HAKKERAGHOXDDR
|
8.7 | IC50 | 4 | — | |
KVXGDBDRJBDLPL
|
8.7 | IC50 | 2 | — | |
PVFBWXXUVZTKAZ
|
8.7 | IC50 | 2 | — | |
DQMLXBWKSFQDIL
|
8.7 | IC50 | 2 | — | |
GWHYIUBNKJSYCV
|
8.6 | IC50 | 2 | — | |
FZEMPTLYQJKICO
|
8.6 | IC50 | 2 | — | |
UUVLZGBRJNIVPH
|
8.6 | IC50 | 2 | — | |
QXIJKQBZACKAMG
|
8.6 | Ki | 2 | — | |
XFNDMVROQNGSOY
|
8.6 | IC50 | 2 | — | |
MWULMTACIBZPGN
|
8.6 | IC50 | 8 | — | |
AIMNRLCNWYRUPJ
|
8.5 | IC50 | 4 | Yes | |
FVFURMJFTAJXRH
|
8.5 | IC50 | 3 | — | |
JCLKKRZMUZBICB
|
8.5 | Ki | 2 | — | |
JFLDPXNTPNHXDV
|
8.5 | IC50 | 2 | — | |
KFIBFLUHCJZUTE
|
8.5 | IC50 | 3 | — | |
KQTXWKJKIOAAAJ
|
8.5 | IC50 | 2 | — | |
MNKSLZNPCRRMKJ
|
8.5 | IC50 | 2 | — | |
OKRHAYBIIRGRNK
|
8.5 | IC50 | 2 | — | |
YIKZESIGFJDKFD
|
8.5 | IC50 | 2 | — | |
ZWAQGKCYZQHRHG
|
8.5 | IC50 | 2 | — | |
NLAHHDDTQFVMAG
|
8.5 | IC50 | 2 | — | |
ZOMSYDARYOMDQY
|
8.5 | Ki | 2 | — | |
BEVTZBDUQNCQFB
|
8.5 | IC50 | 2 | — | |
JFJGUHDHENWREH
|
8.5 | IC50 | 2 | — | |
PHWDAICGTWFRGW
|
8.5 | IC50 | 2 | — | |
SZYIKBVCDSTRPX
|
8.5 | IC50 | 2 | — | |
AGEXLZJKWUQKHA
|
8.4 | IC50 | 2 | — | |
AQUDLJKDUONUMG
|
8.4 | IC50 | 2 | — | |
PUSSNOHHCKDXMM
|
8.4 | Ki | 2 | — |