Target Details
| UniProt AC | Q99640 |
|---|---|
| Gene Symbol | PKMYT1 |
| Protein Name | Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 42
- Clinical molecules 7
- Avg pChEMBL 7.09
KEGG Pathways (3)
Active Molecules (42)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IFPPYSWJNWHOLQ
|
8.2 | IC50 | 52 | Yes | |
ZCCPLJOKGAACRT
|
8.1 | Kd | 599 | — | |
ARBRHWRTXPWZGN
|
8.1 | IC50 | 5 | — | |
MIMOHMCANSGXIG
|
7.8 | IC50 | 15 | — | |
XSNFPLSUBIEKQI
|
7.7 | IC50 | 3 | — | |
YLWKYFSHDVCZRG
|
7.7 | IC50 | 3 | — | |
QHCDMISXSDBVBY
|
7.6 | IC50 | 2 | — | |
BWIJMUPUXMYUQJ
|
7.5 | IC50 | 2 | — | |
GLMBDKLIDHCXRV
|
7.5 | IC50 | 2 | — | |
KCJCFPWXUBRAII
|
7.5 | IC50 | 2 | — | |
LQVPTJNUZOETOA
|
7.5 | IC50 | 2 | — | |
QZKCNMPFOPTCFJ
|
7.5 | IC50 | 3 | — | |
VJZGJJHEEQMXDH
|
7.5 | IC50 | 2 | — | |
XNDTVGPOUOXLTI
|
7.5 | IC50 | 2 | — | |
KBWZVVPCJMAFMN
|
7.5 | IC50 | 3 | — | |
SLCFEJAMCRLYRG
|
7.5 | IC50 | 8 | Yes | |
VAARYSWULJUGST
|
7.4 | Ki | 119 | Yes | |
HDTPGKBMQBCWBG
|
7.2 | IC50 | 2 | — | |
MWKSRKSEWLRPBL
|
7.2 | Kd | 1075 | — | |
CCLATZMUQLEESJ
|
7.2 | IC50 | 2 | — | |
ZHMCGBRGDVCXLS
|
7.2 | IC50 | 5 | — | |
RHLCWIADKMKGBA
|
7.1 | IC50 | 2 | — | |
AMSYYFVSGWPACL
|
7.1 | IC50 | 2 | — | |
AKHLCKMEVWGDGL
|
7.0 | Ki | 4 | — | |
WHYJZCBTMCZRNS
|
7.0 | IC50 | 2 | — | |
OWMPVUWPRQPSFI
|
6.9 | IC50 | 2 | — | |
OUKYUETWWIPKQR
|
6.9 | IC50 | 31 | Yes | |
ZBNZXTGUTAYRHI
|
6.9 | Kd | 102 | Yes | |
NQHLFCVNEBJHOT
|
6.8 | IC50 | 2 | — | |
VBAYIVBRKSERFP
|
6.7 | Ki | 3 | — | |
BQQPGJQMRMUCFZ
|
6.7 | IC50 | 2 | — | |
BTBRBTRLCBPEQY
|
6.6 | IC50 | 2 | — | |
DUNPLBXFZIMEHK
|
6.6 | IC50 | 2 | — | |
FALZOWANVMDHFY
|
6.6 | IC50 | 2 | — | |
UBPYILGKFZZVDX
|
6.5 | Ki | 130 | Yes | |
YCLIWTLPTXAGPQ
|
6.3 | Kd | 3 | — | |
PDXLFGGSCODVJA
|
6.3 | Ki | 3 | — | |
WJVCASAEBZAPDS
|
6.3 | Ki | 2 | — | |
BVHZLDLRNBQWRF
|
6.2 | Ki | 5 | — | |
FPQGOOJFBPSPIZ
|
6.2 | IC50 | 2 | — | |
RVIKUEQPEPKOQM
|
6.1 | IC50 | 2 | — | |
WVUNYSQLFKLYNI
|
6.0 | Kd | 46 | Yes |