Target Details
| UniProt AC | Q99572 |
|---|---|
| Gene Symbol | P2RX7 |
| Protein Name | P2X purinoceptor 7 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF20478 (P2RX7_C) PF00864 (P2X_receptor) |
Summary
- Multi-target molecules 159
- Clinical molecules 0
- Avg pChEMBL 7.06
KEGG Pathways (3)
Active Molecules (159)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZRXFLXAGQMMESA
|
7.3 | IC50 | 2 | — | |
ZVJIOSBCMAOEKO
|
7.3 | IC50 | 2 | — | |
ZWUQOCKDABZQOW
|
7.3 | IC50 | 2 | — | |
ZYNCIRVQJPNTOS
|
7.3 | IC50 | 2 | — | |
NTIPPLUXKZVJHM
|
7.2 | IC50 | 2 | — | |
FJIIZNKTKISOBM
|
7.2 | IC50 | 3 | — | |
MMPAULQSJLVKHP
|
6.9 | IC50 | 3 | — | |
DDYZDHRELNHRNM
|
6.8 | IC50 | 3 | — | |
RJVLFQBBRSMWHX
|
6.8 | IC50 | 2 | — | |
FRVRBHNCPAKNHJ
|
6.8 | IC50 | 3 | — | |
CHILCFMQWMQVAL
|
6.8 | IC50 | 6 | — | |
MIFXBNFNNPOWOG
|
6.8 | IC50 | 3 | — | |
OWGDIPHHKWBGJY
|
6.7 | IC50 | 3 | — | |
YAQRTUXYVQSHDL
|
6.6 | IC50 | 2 | — | |
BESWRIIXEVGTHN
|
6.5 | IC50 | 2 | — | |
CQRVMYXBEDBWRK
|
6.5 | IC50 | 2 | — | |
DJXNRGOBYHTONY
|
6.5 | IC50 | 2 | — | |
DMRKNPNOKKHHGK
|
6.5 | IC50 | 2 | — | |
FGCIGBNLVLTDNM
|
6.5 | IC50 | 2 | — | |
FVDOWIVOMIRGRI
|
6.5 | IC50 | 2 | — | |
GHFUDVAMDRYAKM
|
6.5 | IC50 | 2 | — | |
GOYQGOWROZOAEE
|
6.5 | IC50 | 2 | — | |
GSWAPKOVOZEVRX
|
6.5 | IC50 | 2 | — | |
HGEBTOZUHJCFPT
|
6.5 | IC50 | 2 | — | |
HYJYXNXTCDSEDH
|
6.5 | IC50 | 2 | — | |
KJNJNRKBJCGEIL
|
6.5 | IC50 | 2 | — | |
LIGCUAXRHFCHCD
|
6.5 | IC50 | 2 | — | |
LJFYPZLDGKBVIH
|
6.5 | IC50 | 2 | — | |
MDPSJCJCQNIUMX
|
6.5 | IC50 | 2 | — | |
MLGGONKYUOQNCS
|
6.5 | IC50 | 2 | — | |
OIPFHTDSPCKTSD
|
6.5 | IC50 | 2 | — | |
ORALAQJGVJKTRD
|
6.5 | IC50 | 2 | — | |
OYGOLYUDIIFGEU
|
6.5 | IC50 | 2 | — | |
PAGDEUIXKSZUKR
|
6.5 | IC50 | 2 | — | |
PBCVXOVXFXJEQS
|
6.5 | IC50 | 2 | — | |
PJDGMMHQDJQFSD
|
6.5 | IC50 | 2 | — | |
PPZCGQUVIQDNPL
|
6.5 | IC50 | 2 | — | |
QKROXFAZQDVJQH
|
6.5 | IC50 | 2 | — | |
QUPJJASNZIHKTK
|
6.5 | IC50 | 2 | — | |
REUKACGWWCWKPN
|
6.5 | IC50 | 2 | — | |
SZPRVMAEROLVQD
|
6.5 | IC50 | 2 | — | |
UIYCMEDVXUZDGL
|
6.5 | IC50 | 2 | — | |
USZJYBQKSJDVGU
|
6.5 | IC50 | 2 | — | |
VNZGQQFGKCGUPN
|
6.5 | IC50 | 2 | — | |
WRUQCCISRATVAR
|
6.5 | IC50 | 2 | — | |
WZYMTEJFHFNNGW
|
6.5 | IC50 | 2 | — | |
XGEHFSBNTQEICT
|
6.5 | IC50 | 2 | — | |
XNGBJLAYEZATOX
|
6.5 | IC50 | 2 | — | |
XNHJPRKAGSWPQN
|
6.5 | IC50 | 2 | — | |
LIPWVXLUWLNIBY
|
6.5 | IC50 | 3 | — |