Target Details
| UniProt AC | Q99572 |
|---|---|
| Gene Symbol | P2RX7 |
| Protein Name | P2X purinoceptor 7 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF20478 (P2RX7_C) PF00864 (P2X_receptor) |
Summary
- Multi-target molecules 159
- Clinical molecules 0
- Avg pChEMBL 7.06
KEGG Pathways (3)
Active Molecules (159)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HZABZKYZDQPWMV
|
10.0 | IC50 | 2 | — | |
MUCFYQFETABRSU
|
9.2 | IC50 | 2 | — | |
GRXSJFATZNFEHW
|
8.7 | IC50 | 2 | — | |
FYUUGCZPBDIVNB
|
8.3 | IC50 | 2 | — | |
CJGVMBDHPYMJDI
|
8.2 | IC50 | 2 | — | |
RCRQGABLIRBSJX
|
7.6 | IC50 | 2 | — | |
DIKKTLPJDURHSW
|
7.5 | IC50 | 3 | — | |
DYJDDJVVVMHYEH
|
7.5 | IC50 | 2 | — | |
ACXDVSFQBFMOGD
|
7.3 | IC50 | 2 | — | |
ALBOHFZHNNBACL
|
7.3 | IC50 | 2 | — | |
BBQGQUYUBIGQSH
|
7.3 | IC50 | 2 | — | |
BBQGQUYUBIGQSH
|
7.3 | IC50 | 2 | — | |
BICRBLIUIWVJGT
|
7.3 | IC50 | 2 | — | |
BKGLDWNJYRVNDF
|
7.3 | IC50 | 2 | — | |
BLBOFCVFAJJLMF
|
7.3 | IC50 | 2 | — | |
BSZBTMYXYUODRZ
|
7.3 | IC50 | 2 | — | |
CNTRWIPVLALTDN
|
7.3 | IC50 | 2 | — | |
DZPFVUSVHAVVJR
|
7.3 | IC50 | 2 | — | |
DZPFVUSVHAVVJR
|
7.3 | IC50 | 2 | — | |
DZUUFEFOAJILJT
|
7.3 | IC50 | 2 | — | |
FJOZGEOEQGSXAW
|
7.3 | IC50 | 2 | — | |
FVDOWIVOMIRGRI
|
7.3 | IC50 | 2 | — | |
FVDOWIVOMIRGRI
|
7.3 | IC50 | 2 | — | |
FVDOWIVOMIRGRI
|
7.3 | IC50 | 2 | — | |
GGDYUQIVEMLAOC
|
7.3 | IC50 | 2 | — | |
GGJAAUYAOVPEKL
|
7.3 | IC50 | 2 | — | |
GNVRZHHSFIRPCQ
|
7.3 | IC50 | 2 | — | |
HKIPQWVBOHKCFR
|
7.3 | IC50 | 2 | — | |
HMQCQONQOWJVFE
|
7.3 | IC50 | 2 | — | |
HYJYXNXTCDSEDH
|
7.3 | IC50 | 2 | — | |
IEYUNSWQJICCMF
|
7.3 | IC50 | 2 | — | |
IFBFEVQYBARLBL
|
7.3 | IC50 | 2 | — | |
IIFHYBOYNBPFNR
|
7.3 | IC50 | 2 | — | |
INLBEFOLKKUJOC
|
7.3 | IC50 | 2 | — | |
JEYNBLCSBRFKTN
|
7.3 | IC50 | 2 | — | |
JFQOYWWBQIMYDO
|
7.3 | IC50 | 2 | — | |
JGKPQHVZFCKKIN
|
7.3 | IC50 | 2 | — | |
JRKCRSUXXRTIFW
|
7.3 | IC50 | 2 | — | |
JVKPUMLFVNUGFI
|
7.3 | IC50 | 2 | — | |
KYOXPHAUUKIAKS
|
7.3 | IC50 | 2 | — | |
LIIKQOMTYSBGAC
|
7.3 | IC50 | 2 | — | |
LIWOJUJKVLFKLS
|
7.3 | IC50 | 2 | — | |
LLBDMFJIXKFZFS
|
7.3 | IC50 | 2 | — | |
LXGYUFFRYJZLAY
|
7.3 | IC50 | 2 | — | |
LZMOSSPPMWPJOX
|
7.3 | IC50 | 2 | — | |
MDPSJCJCQNIUMX
|
7.3 | IC50 | 2 | — | |
MEPUDURFSDHOKI
|
7.3 | IC50 | 2 | — | |
MFTWCPAPYQQCLJ
|
7.3 | IC50 | 2 | — | |
MFTWCPAPYQQCLJ
|
7.3 | IC50 | 2 | — | |
MGVADBUYXGVLGL
|
7.3 | IC50 | 2 | — |