Target Details
| UniProt AC | Q99571 |
|---|---|
| Gene Symbol | P2RX4 |
| Protein Name | P2X purinoceptor 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00864 (P2X_receptor) |
Summary
- Multi-target molecules 16
- Clinical molecules 0
- Avg pChEMBL 6.61
KEGG Pathways (3)
Active Molecules (16)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DDYZDHRELNHRNM
|
7.4 | IC50 | 3 | — | |
LQZBDVDATBCNNN
|
7.3 | Ki | 3 | — | |
MIFXBNFNNPOWOG
|
7.3 | IC50 | 3 | — | |
NXDGLRGDIKDWIF
|
6.9 | IC50 | 3 | — | |
CHILCFMQWMQVAL
|
6.8 | IC50 | 6 | — | |
FRVRBHNCPAKNHJ
|
6.8 | IC50 | 3 | — | |
LIPWVXLUWLNIBY
|
6.8 | IC50 | 3 | — | |
FIAFUQMPZJWCLV
|
6.8 | Ki | 3 | — | |
OWGDIPHHKWBGJY
|
6.7 | IC50 | 3 | — | |
IHHXPMMIRSLYRE
|
6.3 | IC50 | 3 | — | |
OAMVIBKEICGPKK
|
6.3 | IC50 | 2 | — | |
FJIIZNKTKISOBM
|
6.2 | IC50 | 3 | — | |
GTIRCXWYMTWWRW
|
6.1 | IC50 | 4 | — | |
MXSCITZYHDRLLP
|
6.0 | IC50 | 3 | — | |
RCRQGABLIRBSJX
|
6.0 | IC50 | 2 | — | |
DYJDDJVVVMHYEH
|
6.0 | IC50 | 2 | — |