Target Details
| UniProt AC | Q99558 |
|---|---|
| Gene Symbol | MAP3K14 |
| Protein Name | Mitogen-activated protein kinase kinase kinase 14 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 224
- Clinical molecules 0
- Avg pChEMBL 8.67
KEGG Pathways (13)
- Alcoholic liver disease
- Apoptosis
- C-type lectin receptor signaling pathway
- Chemical carcinogenesis - reactive oxygen species
- Epithelial cell signaling in Helicobacter pylori infection
- Epstein-Barr virus infection
- Human T-cell leukemia virus 1 infection
- Intestinal immune network for IgA production
- MAPK signaling pathway
- NF-kappa B signaling pathway
- Osteoclast differentiation
- T cell receptor signaling pathway
- TNF signaling pathway
Associated Diseases (1)
Active Molecules (224)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ANKQIJATDOANHF
|
7.0 | Ki | 2 | — | |
FPINDZMLPPFGBN
|
6.8 | Ki | 2 | — | |
DGLFSNZWRYADFC
|
6.8 | IC50 | 12 | — | |
ICDRBJJBVQGHAV
|
6.8 | Ki | 2 | — | |
DCUSCHYHFUKBTL
|
6.7 | Ki | 2 | — | |
QTXIZTUQLFYMNF
|
6.6 | Ki | 2 | — | |
CLVARCBGXGKOMT
|
6.6 | Ki | 2 | — | |
ATUUNJCZCOMUKD
|
6.6 | IC50 | 7 | — | |
WTNAUUFHNUWQGQ
|
6.6 | Ki | 2 | — | |
PGOZOJWRERDXBU
|
6.6 | Ki | 2 | — | |
CMHKURIYUXPNNR
|
6.5 | Ki | 3 | — | |
NXSJMRCTGYTSTK
|
6.5 | Kd | 200 | — | |
FPINDZMLPPFGBN
|
6.4 | Ki | 2 | — | |
OSVUGUHRKMMBSE
|
6.3 | Kd | 170 | — | |
UDOPKESZEISBPX
|
6.3 | Ki | 2 | — | |
MJQUKUIDCUNAAB
|
6.3 | IC50 | 4 | — | |
FZJMLWNUSUKYPU
|
6.2 | Ki | 2 | — | |
HDJJCDBHJXIVLV
|
6.2 | Ki | 2 | — | |
KTPZTVBPMOHXFD
|
6.2 | Ki | 2 | — | |
HZWIAHGTTPPVAC
|
6.2 | Ki | 2 | — | |
WZLQQYUWMGFXDE
|
6.2 | IC50 | 3 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |