Target Details
| UniProt AC | Q99527 |
|---|---|
| Gene Symbol | GPER1 |
| Protein Name | G-protein coupled estrogen receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 9
- Clinical molecules 0
- Avg pChEMBL 8.33
KEGG Pathways (4)
Active Molecules (9)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DAENOLUGFUWJQG
|
10.4 | IC50 | 2 | — | |
DMJJJIYHTDJNMV
|
9.1 | IC50 | 2 | — | |
ZCYXAUDOYRULLH
|
8.9 | IC50 | 2 | — | |
VOXZDWNPVJITMN
|
8.2 | Ki | 8 | — | |
NWYBHLVVGGFXBM
|
7.8 | Ki | 2 | — | |
LFBIANRJUBEHEF
|
7.8 | Ki | 2 | — | |
ALFPTVYCOSMDFS
|
7.6 | Kd | 3 | — | |
VGRGOPKFKWPQOM
|
7.6 | Ki | 2 | — | |
OSMIWTQKPZDLCF
|
7.5 | Ki | 2 | — |