Target Details
| UniProt AC | Q99500 |
|---|---|
| Gene Symbol | S1PR3 |
| Protein Name | Sphingosine 1-phosphate receptor 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 184
- Clinical molecules 0
- Avg pChEMBL 7.32
KEGG Pathways (2)
Active Molecules (184)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CUPKVALESCTXBT
|
6.5 | IC50 | 2 | — | |
FMLHSOGKNHADEE
|
6.5 | Ki | 2 | — | |
MYSPJHRAIVKWQS
|
6.5 | Ki | 2 | — | |
PGLFYYYVMFEVNN
|
6.5 | IC50 | 4 | — | |
PGLFYYYVMFEVNN
|
6.5 | IC50 | 4 | — | |
NOMBGCXWXBTHTO
|
6.5 | IC50 | 4 | — | |
RFNNVHCCTIWJLY
|
6.5 | IC50 | 4 | — | |
MVIUMKOQNNKAJB
|
6.4 | IC50 | 2 | — | |
WMLSDMINRWPYKX
|
6.4 | IC50 | 3 | — | |
GJSCDTCSBXBNCQ
|
6.4 | IC50 | 3 | — | |
UBEBIMAOSJLCDX
|
6.4 | IC50 | 3 | — | |
FSCOADFARBASQU
|
6.4 | IC50 | 4 | — | |
KRYWDAJMWJBMNZ
|
6.3 | IC50 | 4 | — | |
IHJCKBWPCNFLBM
|
6.3 | IC50 | 5 | — | |
IHJCKBWPCNFLBM
|
6.3 | IC50 | 5 | — | |
NCUVDYUSQOEZTJ
|
6.3 | IC50 | 3 | — | |
JGJDBDVJIUNKFZ
|
6.2 | IC50 | 2 | — | |
LRFKWQGGENFBFO
|
6.2 | Ki | 4 | — | |
GBAYNJCGVHFQTM
|
6.2 | IC50 | 4 | — | |
BPFTXGAARBAJDP
|
6.2 | IC50 | 4 | — | |
BLLBAGSMDDITHA
|
6.2 | IC50 | 4 | — | |
YMBOZHBXRGFOHL
|
6.2 | IC50 | 2 | — | |
CSMQUILOGPIVIK
|
6.1 | IC50 | 2 | — | |
LDWAKTDSZSERFS
|
6.1 | IC50 | 3 | — | |
DMDNERFCUCYCGM
|
6.1 | IC50 | 9 | — | |
KUOMYSKEBPYIAO
|
6.1 | IC50 | 4 | — | |
LKIZLUUZCMZBLW
|
6.0 | IC50 | 2 | — | |
BPANWCJVYBGZFM
|
6.0 | IC50 | 4 | — | |
LSZRFUXALRHLHB
|
6.0 | IC50 | 3 | — | |
LYZKFLGVDKUPAP
|
6.0 | IC50 | 4 | — | |
QGDUQFMYMKUVHT
|
6.0 | IC50 | 3 | — | |
UOLFBZYNLRKEKZ
|
6.0 | IC50 | 2 | — | |
WUCGGZATYNFGIA
|
6.0 | IC50 | 4 | — | |
YTTNOAFOCBYIIG
|
6.0 | IC50 | 4 | — |