Target Details
| UniProt AC | Q99500 |
|---|---|
| Gene Symbol | S1PR3 |
| Protein Name | Sphingosine 1-phosphate receptor 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 184
- Clinical molecules 0
- Avg pChEMBL 7.32
KEGG Pathways (2)
Active Molecules (184)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WDBMBYAFMOKUJU
|
9.4 | IC50 | 4 | — | |
DUYSYHSSBDVJSM
|
9.4 | IC50 | 6 | — | |
JBPVYJJIRRUCJU
|
9.2 | IC50 | 4 | — | |
LVLCOLBUGCDLPB
|
9.0 | IC50 | 4 | — | |
MMKMRZFTPGRQEQ
|
9.0 | IC50 | 4 | — | |
YFWUAIPFVJAYCH
|
8.9 | IC50 | 4 | — | |
KARRQFDDSYYFAE
|
8.7 | IC50 | 4 | — | |
AFPYVDIMHNINIS
|
8.6 | IC50 | 4 | — | |
IYOGKTIRIRHPOH
|
8.6 | IC50 | 6 | — | |
IILANYBHYYNGJK
|
8.6 | IC50 | 5 | — | |
LPFGMPGBYMGNTK
|
8.6 | IC50 | 4 | — | |
PEPDHHDQCCNILN
|
8.4 | IC50 | 4 | — | |
ROTPOJPBVJTWLI
|
8.4 | IC50 | 5 | — | |
ZQHLJZUCUJZZRV
|
8.4 | IC50 | 4 | — | |
TWNDWWAUVXKNMU
|
8.4 | IC50 | 4 | — | |
HMJKTOOFFPXTGY
|
8.3 | IC50 | 4 | — | |
PCBMXZQDEQINJG
|
8.3 | IC50 | 4 | — | |
JJPKCGYTCKVOEU
|
8.3 | IC50 | 4 | — | |
ODKLTWJRUVYDRU
|
8.3 | IC50 | 5 | — | |
DUYSYHSSBDVJSM
|
8.3 | Ki | 5 | — | |
IJFAOCYEADEWAV
|
8.2 | IC50 | 4 | — | |
GHQKYJKUIMNJCW
|
8.2 | IC50 | 4 | — | |
RNDGTSGYNDTFOA
|
8.2 | IC50 | 4 | — | |
JTIPBJDEQFMDSI
|
8.2 | IC50 | 2 | — | |
MJFHVHNIHASYLI
|
8.2 | IC50 | 4 | — | |
KKNUGAMJKIHACQ
|
8.2 | IC50 | 4 | — | |
KLULNXUHMWEEKT
|
8.2 | IC50 | 4 | — | |
LCRADRCUDVEFGB
|
8.2 | IC50 | 4 | — | |
LRFKWQGGENFBFO
|
8.2 | IC50 | 5 | — | |
LRFKWQGGENFBFO
|
8.2 | IC50 | 5 | — | |
JWFPFBZCDCVFBO
|
8.2 | IC50 | 2 | — | |
HXDPHSXYLHIVSE
|
8.1 | IC50 | 4 | — | |
CDEPDWBJGIUHRS
|
8.1 | IC50 | 5 | — | |
BDZJQGMIIWGSHK
|
8.1 | IC50 | 4 | — | |
XTEYPDFMLGCQTR
|
8.1 | IC50 | 2 | — | |
GHGMOTNOPRPKKC
|
8.0 | IC50 | 3 | — | |
MSESTOOFLKUAQK
|
8.0 | IC50 | 2 | — | |
XZWUWZDFEBVUJQ
|
8.0 | IC50 | 4 | — | |
XGFCNYXSOCFJIR
|
8.0 | IC50 | 4 | — | |
IWEBRWJRUHNDER
|
8.0 | IC50 | 2 | — | |
MLCQGSONTFRAOL
|
7.9 | IC50 | 2 | — | |
SHQNRSGKLNMHOS
|
7.9 | IC50 | 4 | — | |
ATXJVJPQVHFGIA
|
7.9 | IC50 | 4 | — | |
GRHKCGSXHAHSFS
|
7.9 | IC50 | 2 | — | |
VEAJEWXYGKUGPH
|
7.9 | IC50 | 4 | — | |
JAMOPMAEOMFXHF
|
7.8 | IC50 | 4 | — | |
QDBJDRNNPPZVNE
|
7.8 | IC50 | 2 | — | |
SUTPHRMIWKXQQH
|
7.8 | IC50 | 2 | — | |
XPZPTGRFTGBSAI
|
7.8 | IC50 | 4 | — | |
YHDAWQLKEJHZMN
|
7.8 | IC50 | 4 | — |