Target Details
| UniProt AC | Q99250 |
|---|---|
| Gene Symbol | SCN2A |
| Protein Name | Sodium channel protein type 2 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) PF24609 (IQ_SCN5A_C) PF06512 (Na_trans_assoc) PF11933 (Na_trans_cytopl) |
Summary
- Multi-target molecules 69
- Clinical molecules 4
- Avg pChEMBL 6.99
KEGG Pathways (1)
Associated Diseases (3)
Active Molecules (69)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KGGQAIGGEXFULW
|
6.3 | IC50 | 3 | — | |
DKGZKTPJOSAWFA
|
6.2 | IC50 | 21 | — | |
NEBUOXBYNAHKFV
|
6.2 | IC50 | 5 | — | |
QVZCXCJXTMIDME
|
6.2 | IC50 | 4 | — | |
SMANXXCATUTDDT
|
6.2 | IC50 | 25 | Yes | |
GRLGZDKCJLINRL
|
6.2 | IC50 | 2 | — | |
CQIXHVVDGNOBRL
|
6.2 | IC50 | 2 | — | |
CAFOIGUDKPQBIO
|
6.1 | IC50 | 3 | — | |
RMEDXOLNCUSCGS
|
6.1 | IC50 | 17 | Yes | |
PHSYVYPNRCSHQN
|
6.1 | IC50 | 3 | — | |
UIEATEWHFDRYRU
|
6.1 | IC50 | 8 | — | |
FXTBLDWXLZMPPV
|
6.0 | IC50 | 3 | — | |
HBNPJJILLOYFJU
|
6.0 | IC50 | 21 | — | |
DMUGWPYKKXFQFR
|
6.0 | IC50 | 2 | — | |
HMXDWDSNPRNUKI
|
6.0 | Ki | 72 | — | |
JJCFRYNCJDLXIK
|
6.0 | IC50 | 25 | Yes | |
MDLXULGUOHLVMN
|
6.0 | IC50 | 2 | — | |
VYANEYBOMGSJQI
|
6.0 | IC50 | 2 | — | |
XUEHBVFEQMVDHJ
|
6.0 | IC50 | 2 | — |