Target Details
| UniProt AC | Q99250 |
|---|---|
| Gene Symbol | SCN2A |
| Protein Name | Sodium channel protein type 2 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) PF24609 (IQ_SCN5A_C) PF06512 (Na_trans_assoc) PF11933 (Na_trans_cytopl) |
Summary
- Multi-target molecules 69
- Clinical molecules 4
- Avg pChEMBL 6.99
KEGG Pathways (1)
Associated Diseases (3)
Active Molecules (69)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BJJIKPMJNDTIHW
|
11.2 | IC50 | 3 | — | |
NLTQZTZBFNPMDH
|
9.7 | IC50 | 3 | — | |
RPQXVSUAYFXFJA
|
9.0 | IC50 | 8 | — | |
GFDXIUXAFNREKM
|
8.7 | IC50 | 6 | — | |
WSPHMGORSRQULF
|
8.6 | IC50 | 6 | — | |
CYBITNCPJFQMIJ
|
8.4 | IC50 | 5 | — | |
XUCXIMYTIQZZHZ
|
8.2 | IC50 | 5 | — | |
FPERPEQIXLOVIK
|
8.2 | IC50 | 5 | — | |
DPIPLAYFRAXNRK
|
8.0 | IC50 | 3 | — | |
XQUOWYVEKSXNET
|
7.9 | Kd | 3 | — | |
KLWKJFRXLGLTIH
|
7.9 | IC50 | 4 | — | |
CFMYXEVWODSLAX
|
7.8 | IC50 | 8 | — | |
DPGOQYYAHWEROP
|
7.8 | IC50 | 5 | — | |
LYTCVQQGCSNFJU
|
7.8 | IC50 | 3 | — | |
PTCBNPULJWGSML
|
7.7 | IC50 | 9 | — | |
WPLZOHYVBARFAX
|
7.5 | IC50 | 2 | — | |
GFSUVQOECDPIQJ
|
7.5 | IC50 | 4 | — | |
SXOAHIZWCZOILH
|
7.4 | IC50 | 9 | — | |
KTUKIQYULOKPOV
|
7.3 | IC50 | 4 | — | |
DDGYZFJJKXLJOG
|
7.3 | IC50 | 2 | — | |
YVUQSNJEYSNKRX
|
7.3 | IC50 | 36 | — | |
XOAUGYVLRSCGBG
|
7.2 | IC50 | 8 | — | |
KYBPOTYVFWNSGS
|
7.2 | Kd | 8 | — | |
ANGUVPSJNSWBFO
|
7.2 | IC50 | 4 | — | |
IVBTXSATVJWRLA
|
7.2 | IC50 | 2 | — | |
FQRONRPRMDEQNS
|
7.0 | IC50 | 2 | — | |
HJTNQQWICWEECK
|
7.0 | IC50 | 3 | — | |
MLDMXXWILKZITA
|
7.0 | IC50 | 2 | — | |
ZYSCOUXLBXGGIM
|
6.9 | IC50 | 9 | — | |
DFBDAHMZXJYZJG
|
6.9 | IC50 | 7 | — | |
JJCBTWUQVASSGZ
|
6.9 | IC50 | 2 | — | |
VOJFVKGTRNXOTJ
|
6.9 | IC50 | 4 | — | |
KQQXPTRMUYKUIC
|
6.8 | Kd | 8 | — | |
KUEGRSXKAHKHIA
|
6.8 | IC50 | 5 | — | |
ODABGVBBVPDXSL
|
6.7 | IC50 | 2 | — | |
UUJCWXBORMXXGI
|
6.7 | IC50 | 2 | — | |
URSQNPPONHUJDL
|
6.6 | IC50 | 3 | — | |
ALYSSPGOUMAGSF
|
6.6 | IC50 | 5 | — | |
RDOIQAHITMMDAJ
|
6.6 | IC50 | 13 | — | |
FVGGAZKZIUTNLQ
|
6.6 | IC50 | 5 | — | |
WPYGCZCMGMVGNO
|
6.5 | IC50 | 4 | — | |
IFFPICMESYHZPQ
|
6.5 | IC50 | 4 | — | |
OWKCSDFZMUWPDJ
|
6.5 | IC50 | 2 | — | |
KFGUDEORIBZTGM
|
6.4 | IC50 | 2 | — | |
FEVBKJITJDHASC
|
6.4 | IC50 | 3 | — | |
ZAGGUCLXSCVDCK
|
6.4 | IC50 | 2 | — | |
ZUXRUQOEFBOTGF
|
6.4 | IC50 | 4 | — | |
DERZBLKQOCDDDZ
|
6.4 | IC50 | 20 | Yes | |
ONXXBNABQCHJHC
|
6.3 | IC50 | 2 | — | |
GKCBAIGFKIBETG
|
6.3 | IC50 | 10 | — |