Target Details
| UniProt AC | Q96SW2 |
|---|---|
| Gene Symbol | CRBN |
| Protein Name | Protein cereblon |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02190 (LON_substr_bdg) PF03226 (Yippee-Mis18) |
Summary
- Multi-target molecules 219
- Clinical molecules 1
- Avg pChEMBL 7.37
Associated Diseases (1)
Active Molecules (219)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VFZOAPWJMLHQTB
|
6.2 | IC50 | 2 | — | |
CRAUTELYXAAAPW
|
6.2 | IC50 | 2 | — | |
ZXUCGFSMGYJNRI
|
6.2 | IC50 | 2 | — | |
CBGRGVYIMBGCPT
|
6.2 | IC50 | 2 | — | |
ZIHUTMFSSZFOJL
|
6.2 | IC50 | 2 | — | |
QFWGXTYWCUQWLL
|
6.2 | Kd | 2 | — | |
XYXZUBMCEWJOLA
|
6.2 | IC50 | 2 | — | |
XZWLTIJDAOOAOZ
|
6.2 | IC50 | 2 | — | |
FFERLSHFMZMHLG
|
6.2 | IC50 | 2 | — | |
ZWXLEWVWKZSKRA
|
6.2 | IC50 | 2 | — | |
MWMSBQXTHIEBNT
|
6.2 | IC50 | 2 | — | |
IFISVDOJTJUTBK
|
6.1 | IC50 | 2 | — | |
WGMHCOALNRTCSZ
|
6.1 | IC50 | 2 | — | |
VVOJECSTVKGBLZ
|
6.1 | IC50 | 3 | — | |
HJIALHKCRPBMOA
|
6.1 | IC50 | 2 | — | |
PWBHUSLMHZLGRN
|
6.1 | IC50 | 2 | — | |
DIFUZJAOBZHDGQ
|
6.1 | IC50 | 2 | — | |
RSNPAKAFCAAMBH
|
6.1 | IC50 | 8 | — | |
LBUSZCRLDPVESA
|
6.0 | IC50 | 2 | — |