Target Details
| UniProt AC | Q96SW2 |
|---|---|
| Gene Symbol | CRBN |
| Protein Name | Protein cereblon |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02190 (LON_substr_bdg) PF03226 (Yippee-Mis18) |
Summary
- Multi-target molecules 219
- Clinical molecules 1
- Avg pChEMBL 7.37
Associated Diseases (1)
Active Molecules (219)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UYLCMFFNTCBIBW
|
7.0 | IC50 | 2 | — | |
AIOCFZJGGGEWDK
|
7.0 | IC50 | 2 | — | |
DGDYTCIJBXSVPQ
|
7.0 | IC50 | 2 | — | |
KTEIFNKAUNYNJU
|
7.0 | IC50 | 114 | — | |
XWKQZYOSWGEGIH
|
7.0 | IC50 | 9 | — | |
ZTOYAGORZQZBCF
|
7.0 | IC50 | 2 | — | |
LKEGXJXRNBALBV
|
6.9 | IC50 | 2 | — | |
DUXOGWVIPNJZCP
|
6.9 | Ki | 2 | — | |
CTBFCHXDKXTELK
|
6.8 | IC50 | 2 | — | |
PUEJOCVNXNAMGP
|
6.8 | IC50 | 2 | — | |
JPHZXDBBLIMTNU
|
6.8 | IC50 | 2 | — | |
BEYPVZLSMWIZRD
|
6.8 | IC50 | 4 | — | |
VEVMVFJHHBEQSP
|
6.8 | IC50 | 3 | — | |
UVSMNLNDYGZFPF
|
6.8 | IC50 | 7 | — | |
CNTYYHGBNSQNOR
|
6.8 | IC50 | 2 | — | |
GOTYRUGSSMKFNF
|
6.8 | IC50 | 6 | — | |
IQZLAXNGIATBBF
|
6.8 | IC50 | 3 | — | |
CTQCRJBAHKVGBK
|
6.7 | IC50 | 3 | — | |
HFUNVIYZQZDQCS
|
6.7 | IC50 | 2 | — | |
JMGLSIAOGZDKNZ
|
6.7 | IC50 | 2 | — | |
GHFSHUWOKKVDBF
|
6.7 | IC50 | 2 | — | |
BANRYGZZIMCKNA
|
6.7 | IC50 | 2 | — | |
BYYNQPPTKWNBOG
|
6.7 | Kd | 2 | — | |
IICWMVJMJVXCLY
|
6.6 | IC50 | 2 | — | |
YJSLNCQHRATHFV
|
6.6 | IC50 | 2 | — | |
FSFTZMITKCNGSR
|
6.6 | IC50 | 2 | — | |
CZSOTEJPRKEDGI
|
6.6 | IC50 | 2 | — | |
PEAFNQVFNPFMJQ
|
6.6 | IC50 | 3 | — | |
UEJJHQNACJXSKW
|
6.6 | IC50 | 2 | — | |
KNHZIKBDHRXJHX
|
6.5 | IC50 | 3 | — | |
STPAWIJDTOCXOB
|
6.5 | IC50 | 2 | — | |
OZXPYGFCMJVQLS
|
6.5 | IC50 | 2 | — | |
SPGWKNITNYHIGX
|
6.5 | IC50 | 2 | — | |
WXSOTMXNHJTFKS
|
6.5 | IC50 | 2 | — | |
OXMXTNDWZBEXAL
|
6.5 | Kd | 2 | — | |
LVHBPJYWOSHALG
|
6.5 | IC50 | 2 | — | |
CXTCUKJCQLYMGZ
|
6.5 | IC50 | 2 | — | |
JQUNMWPNAPLWEB
|
6.5 | IC50 | 2 | — | |
SETFNECMODOHTO
|
6.4 | IC50 | 17 | Yes | |
ZBXHNCURDISBRO
|
6.4 | IC50 | 2 | — | |
HJKHARHYGJCYLQ
|
6.4 | IC50 | 2 | — | |
ZUODKONSNNHSAJ
|
6.3 | IC50 | 7 | — | |
SVADXQXVQIZUOT
|
6.3 | IC50 | 3 | — | |
CMOUKMZMDSDCLM
|
6.3 | IC50 | 2 | — | |
GVWBZLKKNJQQQV
|
6.3 | IC50 | 2 | — | |
MPQLCQKBYRSPNA
|
6.3 | IC50 | 2 | — | |
WFFXSERDNVLVGO
|
6.3 | IC50 | 2 | — | |
CTPAIHOLMQBFAW
|
6.3 | Kd | 2 | — | |
KXEXROVTOHCVHU
|
6.2 | IC50 | 2 | — | |
MXJZNPWGQKNANB
|
6.2 | IC50 | 2 | — |