Target Details
| UniProt AC | Q96SW2 |
|---|---|
| Gene Symbol | CRBN |
| Protein Name | Protein cereblon |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02190 (LON_substr_bdg) PF03226 (Yippee-Mis18) |
Summary
- Multi-target molecules 219
- Clinical molecules 1
- Avg pChEMBL 7.37
Associated Diseases (1)
Active Molecules (219)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YTINZZFBHWSAGL
|
7.5 | IC50 | 2 | — | |
IMDNKQXWGGVELD
|
7.5 | IC50 | 3 | — | |
JDHXUMABFAVKIZ
|
7.5 | Kd | 2 | — | |
GUKINEBETXGZNQ
|
7.5 | IC50 | 2 | — | |
JCFHQNJZGSNYNS
|
7.5 | IC50 | 2 | — | |
RCRVGNCDVAROTP
|
7.5 | Kd | 2 | — | |
WJAYJAKMQSJKDW
|
7.5 | IC50 | 3 | — | |
IWBBXOOPRPDUIL
|
7.5 | IC50 | 3 | — | |
SYJHORXMXBZSSH
|
7.5 | IC50 | 3 | — | |
OJBZGRZGVKAUHH
|
7.4 | IC50 | 2 | — | |
HPNZWSHWKWGFMA
|
7.4 | Kd | 2 | — | |
LHUVKOFLIPGEIS
|
7.4 | IC50 | 2 | — | |
VQDRNQBRRSNVOR
|
7.4 | IC50 | 2 | — | |
WCEHIDWONYOKOJ
|
7.4 | IC50 | 3 | — | |
NUWJDBAJYMJUJR
|
7.4 | IC50 | 2 | — | |
QDFNBECATTWIIB
|
7.4 | IC50 | 2 | — | |
ZCOPIRBPZIGHDU
|
7.4 | IC50 | 2 | — | |
FOTJPEPDXXOTQF
|
7.4 | IC50 | 2 | — | |
JGQPZPLJOBHHBK
|
7.4 | IC50 | 3 | — | |
NFCLUGCJOGGYFA
|
7.3 | IC50 | 2 | — | |
BNZBBHXKCFPTND
|
7.3 | IC50 | 2 | — | |
DQGNINFYAAEZKL
|
7.3 | IC50 | 2 | — | |
JFSVSFBLGUFRRC
|
7.3 | IC50 | 2 | — | |
SGHSUUSYNYZHKK
|
7.3 | IC50 | 2 | — | |
VQDRNQBRRSNVOR
|
7.3 | IC50 | 5 | — | |
ZKMPZGMDXOECHS
|
7.3 | IC50 | 2 | — | |
MSGBAYDSSVGFRF
|
7.2 | IC50 | 2 | — | |
BRZGXSNAXRPPFI
|
7.2 | IC50 | 2 | — | |
ODYIWGILJYUPOR
|
7.2 | IC50 | 3 | — | |
CUVRZBKUGKVECT
|
7.2 | IC50 | 2 | — | |
GZJJHSYIBOTFJG
|
7.2 | IC50 | 2 | — | |
IWRKCKJVIQDQDP
|
7.2 | IC50 | 2 | — | |
MTODSPTXTWYZOD
|
7.2 | IC50 | 2 | — | |
TVYQLBCNYFTQLE
|
7.2 | IC50 | 2 | — | |
VGIMJVRUHGWZHN
|
7.2 | IC50 | 2 | — | |
VUZNRWSEUCWVAP
|
7.2 | IC50 | 2 | — | |
XWFRRVWBOAGFII
|
7.2 | IC50 | 2 | — | |
ZEKJFFGYWAEQSY
|
7.2 | IC50 | 2 | — | |
PTJNYVXLFRBJGN
|
7.2 | IC50 | 5 | — | |
JBYQCGLMICPOSQ
|
7.2 | IC50 | 2 | — | |
VNGVKQNBRLGUAS
|
7.1 | IC50 | 2 | — | |
BFZZIGPNZLXGRV
|
7.1 | IC50 | 3 | — | |
QYTHDSMOGXMOPE
|
7.1 | IC50 | 3 | — | |
WAVOEVFKPHUSDB
|
7.1 | IC50 | 3 | — | |
XMPJICVFSDYOEG
|
7.1 | IC50 | 2 | — | |
XYDZHZCXCJNSIB
|
7.0 | IC50 | 3 | — | |
CZCQPLWFGOLPPQ
|
7.0 | IC50 | 2 | — | |
DSWQBZBOYMTXMP
|
7.0 | IC50 | 3 | — | |
QJYCHNPBBAGVAL
|
7.0 | IC50 | 2 | — | |
RIEGJNXDHULIKM
|
7.0 | IC50 | 3 | — |