Target Details
| UniProt AC | Q96SW2 |
|---|---|
| Gene Symbol | CRBN |
| Protein Name | Protein cereblon |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02190 (LON_substr_bdg) PF03226 (Yippee-Mis18) |
Summary
- Multi-target molecules 219
- Clinical molecules 1
- Avg pChEMBL 7.37
Associated Diseases (1)
Active Molecules (219)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XRFXHIPHYYFKHY
|
7.8 | IC50 | 2 | — | |
GMYRPILFZKTDJL
|
7.8 | IC50 | 2 | — | |
IXZOHGPZAQLIBH
|
7.8 | IC50 | 8 | — | |
IPNHNGIFOOJHDF
|
7.8 | IC50 | 3 | — | |
UDRDPSVGVXICRB
|
7.8 | Kd | 2 | — | |
GYXAATIUVYEJQN
|
7.7 | IC50 | 3 | — | |
ALLCHKMKSNIVMZ
|
7.7 | IC50 | 2 | — | |
FTULXIJEWZULEB
|
7.7 | IC50 | 2 | — | |
HFHKKXQGEYYMBR
|
7.7 | IC50 | 2 | — | |
HZJWFCZECUWBMO
|
7.7 | IC50 | 2 | — | |
IMFUTVGKWOXACT
|
7.7 | IC50 | 2 | — | |
IORXXFBCUZOFPD
|
7.7 | IC50 | 2 | — | |
IZELXQMYVJPRBE
|
7.7 | IC50 | 2 | — | |
JAVBYTGNLWEQHR
|
7.7 | IC50 | 2 | — | |
JQXUGPKGNONGRJ
|
7.7 | IC50 | 2 | — | |
KAQZSUHYIKNSMA
|
7.7 | IC50 | 2 | — | |
KOORPPCPKZKWAE
|
7.7 | IC50 | 2 | — | |
LYIYWZRTLQVENK
|
7.7 | IC50 | 2 | — | |
MXVOXRDYHRNSFK
|
7.7 | IC50 | 2 | — | |
NJPKLVFWJMYAQT
|
7.7 | IC50 | 2 | — | |
ONZBQEPGJPEHTB
|
7.7 | IC50 | 2 | — | |
PWTCMKJGIMHBRB
|
7.7 | IC50 | 2 | — | |
PZULGNXWYVWQRV
|
7.7 | IC50 | 2 | — | |
RJRICJLOYKCGKW
|
7.7 | IC50 | 2 | — | |
SXSUZJDEZNZCKM
|
7.7 | IC50 | 2 | — | |
UREMLFMHGHALLS
|
7.7 | IC50 | 2 | — | |
VQSUAUAAFIUPFL
|
7.7 | IC50 | 2 | — | |
WGXCXXWGAWEDSR
|
7.7 | IC50 | 2 | — | |
XKXMVIZLUBDOHD
|
7.7 | IC50 | 2 | — | |
XRILWDIOJGTLRP
|
7.7 | IC50 | 2 | — | |
OIDIVJNMVBHPAC
|
7.7 | IC50 | 2 | — | |
DMMCKRVBNHWAOD
|
7.6 | Kd | 2 | — | |
DOEVCIHTTTYVCC
|
7.6 | IC50 | 2 | — | |
HLDGYGDHHNONSV
|
7.6 | IC50 | 2 | — | |
ITYXEJVELHAHBC
|
7.6 | IC50 | 2 | — | |
ISEZBLQKECWYJU
|
7.6 | IC50 | 2 | — | |
DCGPUMBJALMCLB
|
7.6 | IC50 | 3 | — | |
FURMQZYSFFTQLK
|
7.6 | IC50 | 2 | — | |
HKSBXNVKPFTBIG
|
7.6 | IC50 | 3 | — | |
BTODVRFBCGOZGM
|
7.6 | IC50 | 2 | — | |
MFAVXSAHTAKLRF
|
7.6 | IC50 | 2 | — | |
BHWJDRNVPYLKBM
|
7.6 | IC50 | 2 | — | |
DMMCKRVBNHWAOD
|
7.6 | Kd | 2 | — | |
KBMWMYFFYVRGPQ
|
7.6 | IC50 | 2 | — | |
WSFUNVYDDZKPSU
|
7.6 | IC50 | 3 | — | |
ZIHIUFZFPMILIG
|
7.6 | IC50 | 2 | — | |
KUZXNKUFLRZLHU
|
7.6 | IC50 | 3 | — | |
LPVPLMPEDJZWAQ
|
7.5 | IC50 | 2 | — | |
RWLOGRLTDKDANT
|
7.5 | Kd | 2 | — | |
FKGDRMFOMMYLPA
|
7.5 | IC50 | 3 | — |