Target Details
| UniProt AC | Q96SW2 |
|---|---|
| Gene Symbol | CRBN |
| Protein Name | Protein cereblon |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02190 (LON_substr_bdg) PF03226 (Yippee-Mis18) |
Summary
- Multi-target molecules 219
- Clinical molecules 1
- Avg pChEMBL 7.37
Associated Diseases (1)
Active Molecules (219)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OHGOKRHLLKPKJK
|
9.8 | Kd | 3 | — | |
RBQXHLBIJMHVHI
|
9.7 | Kd | 3 | — | |
UBZCBNADOGDNJL
|
9.7 | Kd | 2 | — | |
FGTNRYWAENEKJL
|
9.6 | Kd | 3 | — | |
JQMIRXOVVPAXPB
|
9.4 | Kd | 2 | — | |
JBMSSKLUVBBAHN
|
9.4 | Kd | 3 | — | |
RMSPJEQBXIFKPD
|
9.3 | IC50 | 3 | — | |
MKHTUOFMIYFSEP
|
9.2 | Kd | 3 | — | |
AJNQGWOQPRWRML
|
8.8 | IC50 | 2 | — | |
ULZLXWZUEUPEEK
|
8.7 | Kd | 2 | — | |
UTYRVEGASOEMJK
|
8.5 | Kd | 2 | — | |
ASTBYSZIHNGCIB
|
8.5 | IC50 | 2 | — | |
MQPRRCLCHOSXND
|
8.5 | IC50 | 3 | — | |
YTQVSNUZNYHPOL
|
8.5 | Kd | 2 | — | |
CKFOAVDINFHZIR
|
8.4 | IC50 | 2 | — | |
TXXHHAICAYYMLP
|
8.4 | IC50 | 2 | — | |
WVKNOEMSHFZOMC
|
8.4 | IC50 | 2 | — | |
XBNLPFPGSKOCJV
|
8.4 | Kd | 2 | — | |
HMNJUXRTSGUSFM
|
8.4 | IC50 | 3 | — | |
INCVUGCZQZUSSU
|
8.3 | IC50 | 2 | — | |
FPHKCZOCTJCWAD
|
8.3 | IC50 | 2 | — | |
FXSJJVJXVNFIBU
|
8.3 | IC50 | 2 | — | |
QMWODUXCOTUXJT
|
8.3 | IC50 | 3 | — | |
CKFOAVDINFHZIR
|
8.3 | IC50 | 2 | — | |
RKAFYSIKAVFVPS
|
8.3 | IC50 | 2 | — | |
IWIUHSRVMHYMOY
|
8.2 | IC50 | 2 | — | |
WDZJVWSRFXJQFY
|
8.2 | Kd | 2 | — | |
YJOJMGTVKMABKQ
|
8.2 | IC50 | 2 | — | |
DGVCXMYHBXQNBX
|
8.2 | Kd | 2 | — | |
GSWRJJUJRPXSPR
|
8.1 | IC50 | 3 | — | |
LKEGXJXRNBALBV
|
8.1 | IC50 | 5 | — | |
GVXKUINUYLVQFZ
|
8.1 | IC50 | 2 | — | |
QJVKGYZEXZRQEQ
|
8.1 | IC50 | 2 | — | |
GYDGGFJIHASCKP
|
8.0 | Kd | 2 | — | |
XOHXSACDCDVFJU
|
8.0 | Kd | 2 | — | |
YYQKAYPIEXTSMF
|
8.0 | IC50 | 2 | — | |
CVNPPCKNNCCUNH
|
8.0 | IC50 | 2 | — | |
LBBCBGBNFQQOSZ
|
8.0 | IC50 | 2 | — | |
PQDZPVHUGZGAPV
|
8.0 | IC50 | 2 | — | |
SIVKMVMSQFNJAG
|
7.9 | IC50 | 2 | — | |
NAJLKAMZDMZECA
|
7.9 | IC50 | 2 | — | |
YPKGJVAMXZZNGJ
|
7.9 | IC50 | 2 | — | |
SVAAFCIDSHIIPD
|
7.9 | IC50 | 2 | — | |
KVKRYCAWRGWYNN
|
7.9 | IC50 | 3 | — | |
RKDBBXGRXIYXMB
|
7.9 | IC50 | 2 | — | |
AILRADAXUVEEIR
|
7.8 | IC50 | 75 | — | |
HLZCITRKGRESDX
|
7.8 | IC50 | 2 | — | |
OKISKGIPUPRZPL
|
7.8 | IC50 | 2 | — | |
RFDBAEYXGSDEIK
|
7.8 | IC50 | 3 | — | |
RQGVCBYHXMUZAF
|
7.8 | Kd | 2 | — |