Target Details
| UniProt AC | Q96SB4 |
|---|---|
| Gene Symbol | SRPK1 |
| Protein Name | SRSF protein kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 88
- Clinical molecules 11
- Avg pChEMBL 7.0
KEGG Pathways (1)
Active Molecules (88)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HATNHAMXMKJCEI
|
6.5 | Ki | 9 | — | |
LKUJDAHYLPICSE
|
6.5 | Ki | 24 | — | |
MVJMMLFMPWITEJ
|
6.5 | Ki | 110 | — | |
RJZDECGDCKOHBV
|
6.5 | Ki | 70 | — | |
UEIRKXUBXCSHJE
|
6.5 | Ki | 19 | — | |
XIOOJUQFJYPVLA
|
6.5 | Ki | 17 | — | |
ZQVQTUFEKLITNT
|
6.5 | Ki | 10 | — | |
SEZFNTZQMWJIAI
|
6.4 | Kd | 9 | Yes | |
BNLPAUPVSCPTDM
|
6.4 | Ki | 15 | — | |
HSKVRPZJBMXFDX
|
6.4 | Ki | 20 | — | |
XCHWBXBDZRJVDP
|
6.4 | Ki | 51 | — | |
PIQCTGMSNWUMAF
|
6.4 | Kd | 137 | Yes | |
BIIVYFLTOXDAOV
|
6.3 | Ki | 31 | — | |
VNGYQBMDQMDALH
|
6.3 | Ki | 25 | — | |
BPNUQXPIQBZCMR
|
6.3 | Kd | 83 | Yes | |
NHHQJBCNYHBUSI
|
6.2 | Kd | 220 | — | |
KXPWWMPXNUOYOH
|
6.2 | Ki | 24 | — | |
UMTWTCVTRDYHQQ
|
6.2 | Ki | 56 | — | |
CACMTVGXYAZZNY
|
6.1 | Ki | 11 | — | |
CLEGDJQQHUTCOW
|
6.1 | Ki | 43 | — | |
OPLHMHMCXQXEQG
|
6.1 | Ki | 10 | — | |
OWDRQHVEJIYVOI
|
6.1 | Ki | 47 | — | |
PCQMERRARZKTPW
|
6.1 | Ki | 68 | — | |
DWFGGOFPIISJIT
|
6.0 | IC50 | 3 | — | |
ADMFLILDQJSEIK
|
6.0 | Ki | 72 | — | |
DKSNLQYRZJKYOC
|
6.0 | Ki | 51 | — | |
FUMCKNCUEAQHCV
|
6.0 | Ki | 103 | — | |
GCYXEGSPUDSZJY
|
6.0 | Ki | 82 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
NHFDRBXTEDBWCZ
|
6.0 | Ki | 41 | — | |
PTVPBWWDGZSEAF
|
6.0 | Ki | 63 | — | |
QQWUGDVOUVUTOY
|
6.0 | Ki | 231 | Yes | |
SBFPHSVZEXSHTL
|
6.0 | Ki | 62 | — | |
SRUYMJRFVGLQDV
|
6.0 | Ki | 37 | — | |
SYLTYCLPHHSEIJ
|
6.0 | Ki | 27 | — | |
UYJNQQDJUOUFQJ
|
6.0 | Ki | 68 | — |