Target Details
| UniProt AC | Q96SB4 |
|---|---|
| Gene Symbol | SRPK1 |
| Protein Name | SRSF protein kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 88
- Clinical molecules 11
- Avg pChEMBL 7.0
KEGG Pathways (1)
Active Molecules (88)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QKYONSSKLFQUAK
|
9.1 | IC50 | 4 | — | |
JINIKYUAUCGQAS
|
8.9 | IC50 | 3 | — | |
XHGQFRKDGWOOTC
|
8.7 | IC50 | 4 | — | |
FFYSPCYXAGHVFZ
|
8.6 | IC50 | 2 | — | |
IVUXRXIUHJUOGX
|
8.6 | IC50 | 2 | — | |
VYUPBBUIPPRDHY
|
8.6 | IC50 | 4 | — | |
QXAZYKBUUHKHCE
|
8.5 | IC50 | 4 | — | |
FXUVMEINVSOBBC
|
8.3 | IC50 | 4 | — | |
BMWIOANJDKPITJ
|
8.3 | IC50 | 4 | — | |
HKSZLNNOFSGOKW
|
8.3 | Kd | 213 | — | |
VURLRACCOCGFDB
|
8.2 | IC50 | 6 | — | |
QDOBOOXEUHHHIB
|
8.2 | IC50 | 2 | — | |
UIARLYUEJFELEN
|
8.0 | Kd | 289 | Yes | |
QPQVHWVHICSFLT
|
7.8 | IC50 | 2 | — | |
WLKNPWYHXQYIKX
|
7.8 | IC50 | 2 | — | |
QCJBCPNAXWXMKR
|
7.8 | IC50 | 2 | — | |
COCWGMSYYWUEJO
|
7.8 | IC50 | 2 | — | |
RSEPBTKMKCSLRW
|
7.7 | IC50 | 2 | — | |
YISMQBFJYDFMAL
|
7.7 | IC50 | 46 | — | |
PXPKETFTEJOGJZ
|
7.6 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
7.6 | IC50 | 408 | — | |
PNKALLUVKOKYHZ
|
7.6 | Ki | 32 | — | |
GHJRTYLEEZPFLY
|
7.5 | IC50 | 2 | — | |
FFTPSTJVKUBPGA
|
7.5 | IC50 | 2 | — | |
SSZBLNIVOGDOJH
|
7.5 | IC50 | 2 | — | |
GXOOVHLYHHEEPZ
|
7.5 | IC50 | 2 | — | |
TWKWEBMGDALHPN
|
7.5 | IC50 | 9 | — | |
CDJFJOKODBBMBI
|
7.4 | IC50 | 2 | — | |
XZXHXSATPCNXJR
|
7.4 | Kd | 165 | Yes | |
GXGUVSXXUOACEX
|
7.4 | IC50 | 2 | — | |
OWRXHGAFWZFFCW
|
7.4 | Ki | 113 | — | |
OYONTEXKYJZFHA
|
7.4 | Kd | 69 | Yes | |
BMGQWWVMWDBQGC
|
7.4 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
7.4 | Kd | 91 | Yes | |
WBFJDKLBAAHKIL
|
7.4 | IC50 | 3 | — | |
KDGFLJKFZUIJMX
|
7.3 | IC50 | 10 | — | |
ALLIMXLDTJFWHR
|
7.3 | IC50 | 2 | — | |
YYLKKYCXAOBSRM
|
7.3 | Kd | 191 | — | |
GNVPRIZIWGZTEE
|
7.2 | IC50 | 2 | — | |
BSFNGHCTZDCQBF
|
7.1 | Ki | 93 | — | |
GCIKSSRWRFVXBI
|
7.1 | Kd | 109 | Yes | |
FPQHXFMYXQZPSV
|
7.0 | Ki | 23 | — | |
VVHBABQYLQVCFE
|
7.0 | IC50 | 2 | — | |
LYADGAGFYYXXIO
|
6.8 | IC50 | 82 | — | |
GFOMFROIIBQABZ
|
6.8 | Ki | 7 | — | |
JOOXLOJCABQBSG
|
6.8 | Kd | 139 | — | |
GHMRUNOHAHJNNA
|
6.7 | Ki | 29 | — | |
MIKAKZKNMYZLDX
|
6.7 | Ki | 42 | — | |
WINHZLLDWRZWRT
|
6.6 | Kd | 201 | Yes | |
AOFJRBMLTUGMMP
|
6.5 | Ki | 12 | — |