Target Details
| UniProt AC | Q96S53 |
|---|---|
| Gene Symbol | TESK2 |
| Protein Name | Dual specificity testis-specific protein kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 11
- Clinical molecules 0
- Avg pChEMBL 7.05
Active Molecules (11)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZCCPLJOKGAACRT
|
9.1 | Kd | 599 | — | |
WVXNSAVVKYZVOE
|
8.7 | Kd | 92 | — | |
MWKSRKSEWLRPBL
|
8.5 | Kd | 1075 | — | |
JUUFLLKHNYWHKP
|
7.8 | Kd | 12 | — | |
WUCYRTXFXRZKSV
|
6.6 | IC50 | 4 | — | |
RYXLLTGGHCFCFK
|
6.4 | IC50 | 3 | — | |
ZEMLGPJIQJHESM
|
6.4 | IC50 | 3 | — | |
NSNKKSURBOMEKE
|
6.2 | IC50 | 3 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |