Target Details
| UniProt AC | Q96RR4 |
|---|---|
| Gene Symbol | CAMKK2 |
| Protein Name | Calcium/calmodulin-dependent protein kinase kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 81
- Clinical molecules 13
- Avg pChEMBL 7.43
KEGG Pathways (7)
Active Molecules (81)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BMGQWWVMWDBQGC
|
7.1 | Kd | 91 | Yes | |
OYONTEXKYJZFHA
|
7.1 | Kd | 69 | Yes | |
ZCCPLJOKGAACRT
|
7.1 | Kd | 599 | — | |
AILRADAXUVEEIR
|
7.1 | IC50 | 75 | — | |
NOMBUNHXDWBICV
|
7.1 | Ki | 11 | — | |
UHSGKZKFUUFRPH
|
7.0 | IC50 | 4 | — | |
MYKOWOGZBMOVBJ
|
6.9 | IC50 | 9 | — | |
DKZYXHCYPUVGAF
|
6.9 | Kd | 112 | — | |
DYNHJHQFHQTFTP
|
6.9 | Kd | 38 | — | |
CPATWHLHNLJLTB
|
6.8 | IC50 | 2 | — | |
JZTOUVBEZONDKA
|
6.8 | Ki | 80 | — | |
PIQCTGMSNWUMAF
|
6.8 | Ki | 137 | Yes | |
UBVFQVJPQKNVPY
|
6.7 | IC50 | 2 | — | |
SXNJFOWDRLKDSF
|
6.7 | Kd | 8 | — | |
DPRNXTSMYVCYLJ
|
6.7 | IC50 | 13 | — | |
KSFDVNIKNYXUIP
|
6.7 | IC50 | 3 | — | |
GZZXEPJJXLJJEJ
|
6.7 | IC50 | 2 | — | |
ODPGGGTTYSGTGO
|
6.7 | Kd | 153 | — | |
MZDKLVOWGIOKTN
|
6.5 | Ki | 80 | — | |
BIIVYFLTOXDAOV
|
6.4 | Kd | 29 | — | |
BIIVYFLTOXDAOV
|
6.4 | Kd | 82 | Yes | |
YYLKKYCXAOBSRM
|
6.3 | Kd | 191 | — | |
DUZMKFLMNMTYDM
|
6.3 | IC50 | 4 | — | |
XKFTZKGMDDZMJI
|
6.3 | Kd | 64 | Yes | |
WINHZLLDWRZWRT
|
6.2 | Ki | 66 | — | |
CWJLAVRXVFHDSJ
|
6.2 | IC50 | 13 | — | |
BPNUQXPIQBZCMR
|
6.1 | Kd | 83 | Yes | |
UBPYILGKFZZVDX
|
6.1 | Kd | 130 | Yes | |
ZZSBPGIGIUFJRA
|
6.1 | Kd | 46 | — | |
XZXHXSATPCNXJR
|
6.0 | Kd | 165 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — |