Target Details
| UniProt AC | Q96RR4 |
|---|---|
| Gene Symbol | CAMKK2 |
| Protein Name | Calcium/calmodulin-dependent protein kinase kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 81
- Clinical molecules 13
- Avg pChEMBL 7.43
KEGG Pathways (7)
Active Molecules (81)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
9.8 | Kd | 408 | — | |
HKSZLNNOFSGOKW
|
9.8 | Kd | 213 | — | |
HKSZLNNOFSGOKW
|
9.7 | Ki | 118 | — | |
OWRXHGAFWZFFCW
|
8.9 | Ki | 113 | — | |
UYJNQQDJUOUFQJ
|
8.9 | Ki | 68 | — | |
PQNZVSVIDDXJQO
|
8.8 | IC50 | 3 | — | |
KOZFSFOOLUUIGY
|
8.7 | Ki | 26 | — | |
HOQCCNALNBIQIM
|
8.7 | IC50 | 2 | — | |
NXSJMRCTGYTSTK
|
8.7 | Kd | 200 | — | |
WVSBGSNVCDAMCF
|
8.5 | IC50 | 4 | — | |
NWXLOTLDKWYYDP
|
8.5 | IC50 | 2 | — | |
OSVUGUHRKMMBSE
|
8.2 | Kd | 170 | — | |
YJRZCHGBUZZOPZ
|
8.1 | IC50 | 2 | — | |
OXICLXLJBMPGTO
|
8.1 | IC50 | 5 | — | |
QQWUGDVOUVUTOY
|
8.0 | Kd | 231 | Yes | |
KASDTXOUSYBOPY
|
7.9 | IC50 | 3 | — | |
QMYPKGGBVVCXIE
|
7.9 | IC50 | 3 | — | |
SOIQVEVFDNZKNF
|
7.9 | IC50 | 3 | — | |
WKCUMDOOJAZCDE
|
7.9 | IC50 | 4 | — | |
ZBAFXJXHSORURK
|
7.9 | IC50 | 4 | — | |
AYDMRHKXWFMUFF
|
7.9 | IC50 | 2 | — | |
FCLPVPNWFDOVKL
|
7.8 | Ki | 11 | — | |
UIARLYUEJFELEN
|
7.8 | Kd | 289 | Yes | |
PSLDQEIGOZTJMS
|
7.8 | IC50 | 3 | — | |
GFADNMXBCPZLOT
|
7.8 | IC50 | 2 | — | |
FXLKAGSPCQYANT
|
7.7 | IC50 | 2 | — | |
SFFKUECRLQXXTN
|
7.7 | IC50 | 3 | — | |
VUTLUBADCGINEP
|
7.7 | IC50 | 3 | — | |
BNYXRPMABDQJJR
|
7.7 | Kd | 5 | — | |
VAYOUJHNIZVWCA
|
7.7 | IC50 | 2 | — | |
XQVVPGYIWAGRNI
|
7.6 | Kd | 34 | — | |
JCMKBZIPVJCSSW
|
7.6 | IC50 | 2 | — | |
JMPYOBZSMKYCFM
|
7.6 | IC50 | 4 | — | |
JTOAKYPOVGNGDU
|
7.6 | IC50 | 3 | — | |
PGBYHFSGSTUFFN
|
7.6 | IC50 | 2 | — | |
SEYKIIXYLAWBHP
|
7.6 | IC50 | 4 | — | |
QLMHELCDKYDUPA
|
7.5 | IC50 | 2 | — | |
PBCZSGKMGDDXIJ
|
7.5 | Kd | 68 | Yes | |
WGWCRXQUBYJTRA
|
7.5 | Ki | 11 | — | |
QFHPSDWMERSJDZ
|
7.5 | IC50 | 4 | — | |
YITXQMHAQVCANR
|
7.5 | IC50 | 3 | — | |
LIHGFLPDHFTNOG
|
7.5 | IC50 | 2 | — | |
YMYOREROCXXANC
|
7.5 | IC50 | 4 | — | |
LIZGTJPPOJGDHW
|
7.5 | IC50 | 2 | — | |
GZYIVQMHOULGOR
|
7.3 | IC50 | 2 | — | |
JWILUIVAYLRFIY
|
7.3 | IC50 | 14 | — | |
KDKUVYLMPJIGKA
|
7.2 | Ki | 91 | Yes | |
OKIHVJIMTWMQNF
|
7.2 | IC50 | 2 | — | |
XJIRZGFXJJLMOT
|
7.2 | IC50 | 2 | — | |
BMGQWWVMWDBQGC
|
7.1 | Kd | 147 | Yes |