Target Details
| UniProt AC | Q96RI1 |
|---|---|
| Gene Symbol | NR1H4 |
| Protein Name | Bile acid receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00104 (Hormone_recep) PF00105 (zf-C4) |
Summary
- Multi-target molecules 16
- Clinical molecules 1
- Avg pChEMBL 8.96
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (16)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AYYWZAJMBFSYQP
|
10.0 | IC50 | 2 | — | |
VGBYMVXRZITCDC
|
9.9 | IC50 | 2 | — | |
IQXGLAOJZLZEGK
|
9.8 | IC50 | 2 | — | |
XULSCZPZVQIMFM
|
9.8 | IC50 | 2 | — | |
PWMAUDHMHOFLLG
|
9.7 | IC50 | 2 | — | |
RYGKFDKOOXWTRF
|
9.7 | IC50 | 2 | — | |
LRMSUSCIZQUFOX
|
9.5 | IC50 | 2 | — | |
HIFUOIYLHIGQEL
|
9.5 | IC50 | 2 | — | |
AWXYVTGPUROLKQ
|
9.4 | IC50 | 2 | — | |
SXDSSOMMAZTTMP
|
9.4 | IC50 | 2 | — | |
SKKDVDAOVWNTOW
|
9.3 | IC50 | 2 | — | |
XFLQIRAKKLNXRQ
|
8.9 | IC50 | 2 | — | |
SMEROWZSTRWXGI
|
7.7 | IC50 | 2 | — | |
XAVJTYOBWCSWFJ
|
7.7 | IC50 | 2 | — | |
IMPXBWVTYSVBEU
|
6.9 | Kd | 2 | — | |
VWUXBMIQPBEWFH
|
6.1 | IC50 | 8 | Yes |