Target Details
| UniProt AC | Q96RI0 |
|---|---|
| Gene Symbol | F2RL3 |
| Protein Name | Proteinase-activated receptor 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 62
- Clinical molecules 0
- Avg pChEMBL 8.17
KEGG Pathways (5)
Active Molecules (62)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UPWRYEAGKLIQQY
|
7.5 | IC50 | 2 | — | |
IMXMVBFSNWACTO
|
7.4 | IC50 | 2 | — | |
NREGDMIGOWLBKQ
|
7.3 | IC50 | 2 | — | |
GMPWJHCKUFHLJE
|
7.3 | IC50 | 2 | — | |
LZKMIVXPFPBCFC
|
7.0 | IC50 | 2 | — | |
UWNZCZNHUPLBBY
|
6.9 | IC50 | 2 | — | |
YPXQVZHMDFVOFI
|
6.8 | IC50 | 2 | — | |
FJAOGFGHTPYADT
|
6.4 | IC50 | 2 | — | |
YYPCMHMJIQOTMJ
|
6.3 | IC50 | 2 | — | |
LPHKQDNIANODOF
|
6.3 | IC50 | 2 | — | |
YHASTZKIWUZWDO
|
6.2 | IC50 | 2 | — | |
VEYNGJJQBIEPNE
|
6.0 | IC50 | 2 | — |