Target Details
| UniProt AC | Q96RI0 |
|---|---|
| Gene Symbol | F2RL3 |
| Protein Name | Proteinase-activated receptor 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 62
- Clinical molecules 0
- Avg pChEMBL 8.17
KEGG Pathways (5)
Active Molecules (62)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RROGCGMHOWNSLD
|
10.1 | IC50 | 2 | — | |
GOQXRFYWUHPILG
|
9.5 | IC50 | 2 | — | |
QGDLVNWXOJELBV
|
9.4 | IC50 | 2 | — | |
BFJWHYCHYOUZLZ
|
9.4 | IC50 | 2 | — | |
PIRVYNOHTBFSEF
|
9.3 | IC50 | 2 | — | |
ZFBVWXYOLVFQGN
|
9.3 | IC50 | 2 | — | |
SRNIWQIVVVDOLO
|
9.2 | IC50 | 2 | — | |
UEPOSULLGAYZQZ
|
9.1 | IC50 | 2 | — | |
KEEBLYWBELVGPQ
|
9.0 | IC50 | 3 | — | |
NUUVIYWKLAQTDU
|
9.0 | IC50 | 2 | — | |
BJIQNZYXWYUXEW
|
9.0 | IC50 | 2 | — | |
MINMDCMSHDBHKG
|
9.0 | IC50 | 2 | — | |
FFXFDFRJDPWERF
|
9.0 | IC50 | 2 | — | |
GFCCZFCZIXBOIU
|
9.0 | IC50 | 2 | — | |
AUHROPMDFWDFRD
|
8.9 | IC50 | 2 | — | |
RACJERJJTUONSE
|
8.9 | IC50 | 2 | — | |
IDEORNGCCVYCFX
|
8.8 | IC50 | 2 | — | |
GZRBIJYGDCLWCQ
|
8.8 | IC50 | 2 | — | |
OLKUSWOEHSSOHD
|
8.8 | IC50 | 2 | — | |
QJDXGILNNBHQDK
|
8.8 | IC50 | 2 | — | |
MVBZVIDGYJOWNV
|
8.7 | IC50 | 2 | — | |
SMSISCIMPYBOQW
|
8.7 | IC50 | 2 | — | |
BKKXFHYCELTMFP
|
8.7 | IC50 | 2 | — | |
KOQWYAURZBRJBF
|
8.7 | IC50 | 2 | — | |
PUHFAUFRLDIBFL
|
8.7 | IC50 | 2 | — | |
IMLVEYAVSNLRRR
|
8.7 | IC50 | 2 | — | |
OLFJSYFEVMJTBF
|
8.7 | IC50 | 2 | — | |
SXPDDHWGSHXZBG
|
8.7 | IC50 | 2 | — | |
LNKZFVATLOPJQY
|
8.6 | IC50 | 2 | — | |
WIJXQXSKKBTTEU
|
8.5 | IC50 | 2 | — | |
LVCJHIUPGAKASO
|
8.5 | IC50 | 2 | — | |
AABZTMRZWJMBNH
|
8.4 | IC50 | 2 | — | |
ZLWUPXBJIJIQJF
|
8.4 | IC50 | 2 | — | |
ZFYDPZVRBWBDPL
|
8.2 | IC50 | 2 | — | |
YGACWBAYURXDEP
|
7.9 | IC50 | 2 | — | |
LSBYGNDYSQKWHF
|
7.8 | IC50 | 2 | — | |
GEOOUXGQTSKLIU
|
7.6 | IC50 | 2 | — | |
SWDKZGZHCMKCKA
|
7.6 | IC50 | 2 | — | |
GBTPSLPMUMGGLO
|
7.6 | IC50 | 2 | — | |
ZRXWJXATIKDMQH
|
7.6 | IC50 | 2 | — | |
VNOAMEZLBNKPPP
|
7.6 | IC50 | 2 | — | |
CXAXQTROOVVLBS
|
7.6 | IC50 | 2 | — | |
QJVPFNRNEFGXGC
|
7.6 | IC50 | 2 | — | |
CANZBHVBEWKJFW
|
7.6 | IC50 | 2 | — | |
NCBXGBVDHSJXGK
|
7.6 | IC50 | 2 | — | |
CXZHQWBVEDJXCG
|
7.6 | IC50 | 2 | — | |
GLZIACYLPINALG
|
7.6 | IC50 | 2 | — | |
YDLUCTVUUDEGBX
|
7.6 | IC50 | 2 | — | |
SBAHBPUZCJUMPW
|
7.5 | IC50 | 2 | — | |
ZJDGGFCBBONCDM
|
7.5 | IC50 | 2 | — |