Target Details
| UniProt AC | Q96Q15 |
|---|---|
| Gene Symbol | SMG1 |
| Protein Name | Serine/threonine-protein kinase SMG1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02260 (FATC) PF00454 (PI3_PI4_kinase) PF15785 (SMG1) PF17229 (SMG1_N) |
Summary
- Multi-target molecules 15
- Clinical molecules 0
- Avg pChEMBL 8.07
KEGG Pathways (1)
Active Molecules (15)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NWQHTOFIQMYFRC
|
10.0 | IC50 | 6 | — | |
RZFJBSIAXYEPBX
|
10.0 | IC50 | 6 | — | |
DTNXNLFOABWGKC
|
9.7 | IC50 | 5 | — | |
YKVXFJUHOCXIAS
|
9.7 | IC50 | 4 | — | |
CICSYFWWWTXRPT
|
8.5 | IC50 | 3 | — | |
CZDONRYGQBBPBK
|
8.5 | IC50 | 4 | — | |
HBLUJJRKHYEUPJ
|
8.2 | IC50 | 4 | — | |
SUIVLXMKJVEBQK
|
8.0 | IC50 | 4 | — | |
FYYYMEMZRSXLIX
|
7.7 | IC50 | 4 | — | |
GCIMHCJOZUYMTH
|
7.6 | IC50 | 3 | — | |
IYNDTACKOAXKBJ
|
7.0 | IC50 | 17 | — | |
MWKSRKSEWLRPBL
|
6.9 | Kd | 1075 | — | |
DGUMNVQVABBBNL
|
6.5 | IC50 | 3 | — | |
GOSZNPGORCKQLX
|
6.5 | IC50 | 3 | — | |
AMGRGTYETFMYTK
|
6.3 | IC50 | 2 | — |