Target Details
| UniProt AC | Q96PY6 |
|---|---|
| Gene Symbol | NEK1 |
| Protein Name | Serine/threonine-protein kinase Nek1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 229
- Clinical molecules 0
- Avg pChEMBL 8.01
Associated Diseases (4)
Active Molecules (229)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LHZSCNHIQYURJR
|
7.2 | IC50 | 2 | — | |
UISKFSKGRDJBFK
|
7.2 | IC50 | 2 | — | |
BAGJPDYVOWKTFN
|
7.2 | IC50 | 2 | — | |
QSTRDZKAPUTJCL
|
7.2 | IC50 | 2 | — | |
IVTXKZOAEFIJGG
|
7.2 | IC50 | 2 | — | |
INSXCHLFWDLFGN
|
7.2 | IC50 | 2 | — | |
CAQDNIUJCQIJSN
|
7.2 | IC50 | 2 | — | |
MBWJUWFANMBYHY
|
7.2 | IC50 | 2 | — | |
HKKPCLDSLIZWJM
|
7.1 | IC50 | 2 | — | |
APIJSFSFSPDPLN
|
7.1 | IC50 | 2 | — | |
OUVMMTWUDVNCFP
|
7.1 | IC50 | 2 | — | |
QBTAZLWMEYVBSX
|
7.1 | IC50 | 2 | — | |
VUEWLORAHCWFHP
|
7.1 | IC50 | 2 | — | |
MMYHBULUVREXPP
|
7.1 | IC50 | 2 | — | |
LGICPSFBCIDMAT
|
7.1 | IC50 | 2 | — | |
OIOUIPSTQHPGEN
|
7.1 | IC50 | 2 | — | |
DNRFMSJVTXHVCU
|
7.1 | IC50 | 2 | — | |
SJVBKIJJPQBWCC
|
7.1 | IC50 | 2 | — | |
JOYSKMLFEFBTPY
|
7.1 | IC50 | 2 | — | |
YKNNQNCGYOGHRS
|
7.0 | IC50 | 2 | — | |
NHHQJBCNYHBUSI
|
6.8 | Kd | 220 | — | |
YPKLAWUGDWZBMV
|
6.8 | IC50 | 2 | — | |
YISMQBFJYDFMAL
|
6.6 | IC50 | 46 | — | |
DZFZXPPHBWCXPQ
|
6.4 | Kd | 12 | — | |
BFSMGDJOXZAERB
|
6.3 | Kd | 33 | — | |
ZEHBZHZMQSHZFI
|
6.2 | IC50 | 2 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |