Target Details
| UniProt AC | Q96PN8 |
|---|---|
| Gene Symbol | TSSK3 |
| Protein Name | Testis-specific serine/threonine-protein kinase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 7
- Clinical molecules 0
- Avg pChEMBL 6.69
Active Molecules (7)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
8.2 | IC50 | 408 | — | |
DGLFSNZWRYADFC
|
7.0 | IC50 | 12 | — | |
OSVUGUHRKMMBSE
|
6.5 | Kd | 170 | — | |
NXSJMRCTGYTSTK
|
6.4 | Kd | 200 | — | |
LZQQEGBCKOIYIP
|
6.4 | IC50 | 4 | — | |
WVYPOHDPGYBAGO
|
6.4 | IC50 | 4 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — |