Target Details
| UniProt AC | Q96PF2 |
|---|---|
| Gene Symbol | TSSK2 |
| Protein Name | Testis-specific serine/threonine-protein kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 29
- Clinical molecules 2
- Avg pChEMBL 6.68
Active Molecules (29)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
8.5 | IC50 | 408 | — | |
QQWUGDVOUVUTOY
|
8.0 | Ki | 231 | Yes | |
FZBVNCFBCNXULH
|
7.5 | IC50 | 18 | — | |
MIKAKZKNMYZLDX
|
7.4 | Ki | 42 | — | |
JSKUWFIZUALZLX
|
7.2 | Ki | 33 | — | |
JZTOUVBEZONDKA
|
7.1 | Ki | 80 | — | |
UMTWTCVTRDYHQQ
|
7.1 | Ki | 56 | — | |
ZGZVRPRSFXRGCF
|
7.1 | Ki | 76 | — | |
OWRXHGAFWZFFCW
|
7.0 | Ki | 113 | — | |
XPHWIERLJBFPFV
|
7.0 | Ki | 69 | — | |
AILRADAXUVEEIR
|
6.9 | IC50 | 75 | — | |
CKVWQORGCCEYHS
|
6.8 | Ki | 50 | — | |
JCFJQIHDZHHMQT
|
6.8 | Ki | 42 | — | |
MVJMMLFMPWITEJ
|
6.7 | Ki | 110 | — | |
RYYNGWLOYLRZLK
|
6.6 | Ki | 104 | — | |
LKUJDAHYLPICSE
|
6.5 | Ki | 24 | — | |
HSKVRPZJBMXFDX
|
6.3 | Ki | 20 | — | |
RJZDECGDCKOHBV
|
6.3 | Ki | 70 | — | |
KTEIFNKAUNYNJU
|
6.2 | Ki | 48 | — | |
WINHZLLDWRZWRT
|
6.2 | Ki | 66 | — | |
ADMFLILDQJSEIK
|
6.1 | Ki | 72 | — | |
BNLPAUPVSCPTDM
|
6.1 | Ki | 15 | — | |
BSFNGHCTZDCQBF
|
6.1 | Ki | 93 | — | |
FLEAYYMORDPWAJ
|
6.1 | Ki | 90 | — | |
OLVBAUVSICCWEJ
|
6.1 | Ki | 39 | — | |
BNSPEWBMGVWZFC
|
6.0 | IC50 | 7 | — | |
OLUKILHGKRVDCT
|
6.0 | Ki | 44 | Yes | |
UOVCGJXDGOGOCZ
|
6.0 | Ki | 59 | — | |
UXUQVXDYXKMCGA
|
6.0 | Ki | 21 | — |