Target Details
| UniProt AC | Q96P20 |
|---|---|
| Gene Symbol | NLRP3 |
| Protein Name | NACHT, LRR and PYD domains-containing protein 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF14484 (FISNA) PF13516 (LRR_6) PF05729 (NACHT) PF17776 (NLRC4_HD2) PF02758 (PYRIN) PF17779 (WHD_NOD2) |
Summary
- Multi-target molecules 16
- Clinical molecules 0
- Avg pChEMBL 7.92
KEGG Pathways (12)
Associated Diseases (6)
Active Molecules (16)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BGHBRFNKKNQTOB
|
9.4 | IC50 | 2 | — | |
XYJKIUDOTQKQBQ
|
9.4 | IC50 | 2 | — | |
UVVZGYXCKGWWCC
|
9.0 | IC50 | 2 | — | |
JEXSOFPQDXJKCO
|
8.6 | IC50 | 2 | — | |
RZADJFPOASAKCT
|
8.3 | IC50 | 2 | — | |
SOZVZFKPLUXVMT
|
8.2 | IC50 | 2 | — | |
HAMGPBKPACGWND
|
8.1 | IC50 | 2 | — | |
NFWAITKLWZRIGK
|
8.0 | Kd | 6 | — | |
XPQDNIYYHPOBPO
|
7.9 | IC50 | 2 | — | |
UZIPRJJBZBJTBL
|
7.7 | IC50 | 2 | — | |
GDAHMFIDUIIGMC
|
7.6 | IC50 | 2 | — | |
JJTXCTVPZBDASI
|
7.5 | IC50 | 2 | — | |
BTNVNDWLDGUCMY
|
7.4 | IC50 | 2 | — | |
XVSWTKVMBWTRFL
|
7.0 | IC50 | 2 | — | |
QTGZVQJHMCFCHW
|
6.5 | IC50 | 2 | — | |
ICUTUKXCWQYESQ
|
6.1 | IC50 | 3 | — |