Target Details
| UniProt AC | Q96NX5 |
|---|---|
| Gene Symbol | CAMK1G |
| Protein Name | Calcium/calmodulin-dependent protein kinase type 1G |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 15
- Clinical molecules 4
- Avg pChEMBL 6.86
KEGG Pathways (4)
Active Molecules (15)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BWBUPDTUXQDHSX
|
9.0 | IC50 | 5 | — | |
PIQCTGMSNWUMAF
|
9.0 | Kd | 137 | Yes | |
HKSZLNNOFSGOKW
|
7.6 | Kd | 408 | — | |
HKSZLNNOFSGOKW
|
7.6 | Kd | 213 | — | |
RZUOCXOYPYGSKL
|
6.9 | Kd | 8 | — | |
XZXHXSATPCNXJR
|
6.6 | Kd | 165 | Yes | |
OSVUGUHRKMMBSE
|
6.5 | Kd | 170 | — | |
NXSJMRCTGYTSTK
|
6.5 | Kd | 200 | — | |
WINHZLLDWRZWRT
|
6.4 | Kd | 201 | Yes | |
NHHQJBCNYHBUSI
|
6.3 | Kd | 220 | — | |
UIARLYUEJFELEN
|
6.3 | Kd | 289 | Yes | |
CTNPALGJUAXMMC
|
6.0 | Kd | 151 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |