Target Details
| UniProt AC | Q96NT5 |
|---|---|
| Gene Symbol | SLC46A1 |
| Protein Name | Proton-coupled folate transporter |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07690 (MFS_1) |
Summary
- Multi-target molecules 34
- Clinical molecules 1
- Avg pChEMBL 7.06
KEGG Pathways (5)
Associated Diseases (1)
Active Molecules (34)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VEKHZPVGFDPVJG
|
8.3 | IC50 | 5 | — | |
JWZBILLJZHUAOY
|
8.2 | IC50 | 5 | — | |
RMEHPWHLFJJYTB
|
8.2 | IC50 | 5 | — | |
UNSSSMUKJOLMJV
|
7.8 | IC50 | 5 | — | |
WMTFSFGBNBUALY
|
7.7 | IC50 | 5 | — | |
BDXBDXZHMOFNOY
|
7.6 | IC50 | 3 | — | |
WGEYLZWUJAEXSI
|
7.3 | IC50 | 2 | — | |
WMBYSCVMFMNUQV
|
7.3 | IC50 | 5 | — | |
ARIQPXNXGFKWNW
|
7.2 | IC50 | 3 | — | |
FSOJIOKMUXQEMI
|
7.2 | IC50 | 5 | — | |
OGSBUKJUDHAQEA
|
7.2 | IC50 | 5 | — | |
STQPVYHCDNSBIJ
|
7.2 | IC50 | 5 | — | |
QLSVPQAGJDLITE
|
7.2 | IC50 | 5 | — | |
CTSPVOIVQCLQLX
|
7.1 | IC50 | 3 | — | |
SIDIEQMDPONVCD
|
7.1 | IC50 | 3 | — | |
WBXPDJSOTKVWSJ
|
7.1 | IC50 | 10 | Yes | |
UPENPAQNDNZZTP
|
7.1 | IC50 | 5 | — | |
IVTVGDXNLFLDRM
|
7.0 | IC50 | 8 | — | |
QXWUFUZJYLBZQF
|
7.0 | IC50 | 3 | — | |
FBOZXECLQNJBKD
|
6.9 | IC50 | 16 | — | |
ADFLVKAWSSGDBU
|
6.9 | Ki | 3 | — | |
JLRJTWXBYRMGEB
|
6.8 | IC50 | 4 | — | |
VMGGIKVXYOZFJO
|
6.8 | IC50 | 4 | — | |
VFYUKZOGWIMWFW
|
6.7 | IC50 | 5 | — | |
STXAYXIUQRNEBG
|
6.7 | IC50 | 3 | — | |
CEPQCJFDTGQKDN
|
6.7 | IC50 | 4 | — | |
CYOOKDIMCAPJGV
|
6.6 | IC50 | 5 | — | |
HPAURQDCTYKMTE
|
6.6 | IC50 | 4 | — | |
UFNWIIALSMNORN
|
6.6 | IC50 | 5 | — | |
FTSMBZFBGMYYIT
|
6.5 | IC50 | 5 | — | |
HQPQAUMWVMDRCN
|
6.5 | IC50 | 3 | — | |
JBVKQLSCSCXKDY
|
6.4 | Ki | 2 | — | |
QNFVXICXLFWABV
|
6.3 | IC50 | 3 | — | |
PNRJTEIZPOHDEE
|
6.1 | IC50 | 2 | — |