Target Details
| UniProt AC | Q96L73 |
|---|---|
| Gene Symbol | NSD1 |
| Protein Name | Histone-lysine N-methyltransferase, H3 lysine-36 specific |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17907 (AWS) PF17982 (C5HCH) PF00628 (PHD) PF23011 (PHD-1st_NSD) PF22908 (PHD_NSD) PF23004 (PHDvar_NSD) PF00855 (PWWP) PF00856 (SET) |
Summary
- Multi-target molecules 5
- Clinical molecules 0
- Avg pChEMBL 6.66
KEGG Pathways (2)
Associated Diseases (1)
Active Molecules (5)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OPJPZRUHVUFNAY
|
6.8 | IC50 | 3 | — | |
NKBVGYWANONFTE
|
6.7 | IC50 | 2 | — | |
DGGOQICQTAGRMC
|
6.7 | IC50 | 3 | — | |
FUEGZWGKKBGDBO
|
6.6 | IC50 | 3 | — | |
WLGCCCLQJAMXCP
|
6.6 | IC50 | 3 | — |